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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
A potent and selective inhibitor for the UBLCP1 proteasome phosphatase.EBI
Indiana University
Characterization of two distinct structural classes of selective aldehyde dehydrogenase 1A1 inhibitors.EBI
Indiana University
Design, synthesis, biochemical studies, cellular characterization, and structure-based computational studies of small molecules targeting the urokinase receptor.EBI
Indiana University
Bicyclic benzofuran and indole-based salicylic acids as protein tyrosine phosphatase inhibitors.EBI
Indiana University
A new glucagon and GLP-1 co-agonist eliminates obesity in rodents.EBI
Indiana University
Amino- and guanidinoacylryanodines: basic ryanodine esters with enhanced affinity for the sarcoplasmic reticulum Ca(2+)-release channel.EBI
Indiana University
Small molecule inhibitors of SHP2 tyrosine phosphatase discovered by virtual screening.EBI
Indiana University
Comprehensive in vitro analysis of voriconazole inhibition of eight cytochrome P450 (CYP) enzymes: major effect on CYPs 2B6, 2C9, 2C19, and 3A.EBI
Indiana University
Structure-Activity Relationship Study of Cannabidiol-Based Analogs as Negative Allosteric Modulators of the μ-Opioid Receptor.EBI
Indiana University
Small-Molecule Cyanamide Pan-TEAD·YAP1 Covalent Antagonists.EBI
Indiana University
Optimization of Truncated Glucagon Peptides to Achieve Selective, High Potency, Full Antagonists.EBI
Indiana University
Pyridyl-alanine as a Hydrophilic, Aromatic Element in Peptide Structural Optimization.EBI
Indiana University
Targeting the HSP60/10 chaperonin systems of Trypanosoma brucei as a strategy for treating African sleeping sickness.EBI
Indiana University
GroEL/ES inhibitors as potential antibiotics.EBI
Indiana University
A biochemical screen for GroEL/GroES inhibitors.EBI
Indiana University
Screening serine/threonine and tyrosine kinase inhibitors for histidine kinase inhibition.EBI
Indiana University
Hydroxamic Acid Compound Having ENPP1 Inhibitory Activity and Use ThereofBDB
Haihe Biopharma
Systems-based design of bi-ligand inhibitors of oxidoreductases: filling the chemical proteomic toolbox.BDB
Triad Therapeutics