Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50036130
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044989((O10eq)-beta-guanidinopropionylryanodine | CHEMBL2...)
Affinity DataIC50: 1.10nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044982(CHEMBL283836 | GLYCYLRYANODINE)
Affinity DataIC50: 1.80nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044986((O10eq)-guanidino acetylryanodine | CHEMBL435362)
Affinity DataIC50: 1.80nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044995((O10eq)-beta-alanylryanodine | CHEMBL282089)
Affinity DataIC50: 2.60nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044993(Benzyloxycarbonyl-glycylryanodine | CHEMBL28383)
Affinity DataIC50: 4.80nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044990((O10eq)-Benzyloxycarbonyl-beta-alanylryanodine | C...)
Affinity DataIC50: 5.90nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044994(Ryanodine | 2,6,9,11,13,14-hexahydroxy-11-isopropy...)
Affinity DataIC50: 6.20nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044991(2,6,9,11,13,14-hexahydroxy-11-isopropyl-7,10-dimet...)
Affinity DataIC50: 8.90nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044987((O10eq)-beta-N,N'-Bis-Benzyloxycarbonyl-guanidinop...)
Affinity DataIC50: 44nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044988(N-methyl ryanodine-succinamidate | CHEMBL432278)
Affinity DataIC50: 49nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044984(Di-Benzyloxycarbonyl-guanidino acetylryanodine | C...)
Affinity DataIC50: 136nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044992((O10eq)-beta-alanyl-anhydro-ryanodine | CHEMBL2826...)
Affinity DataIC50: 149nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044985(ryanodine-hemi-succinate)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044991(2,6,9,11,13,14-hexahydroxy-11-isopropyl-7,10-dimet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Rabbit)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50044991(2,6,9,11,13,14-hexahydroxy-11-isopropyl-7,10-dimet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity for sarcoplasmic reticular calcium release channel (SR CRC) of rabbit skeletal membrane vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed