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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of the minimum PAR4 inhibitor pharmacophore and optimization of a series of 2-methoxy-6-arylimidazo[2,1-b][1,3,4]thiadiazoles.EBI
Vanderbilt University Medical Center
Substituted indoles as selective protease activated receptor 4 (PAR-4) antagonists: Discovery and SAR of ML354.EBI
Northwest Agriculture & Forestry University
Discovery of Two Novel Antiplatelet Clinical Candidates (BMS-986120 and BMS-986141) That Antagonize Protease-Activated Receptor 4.EBI
Bristol-Myers Squibb Research & Early Development
Synthesis and evaluation of novel and potent protease activated receptor 4 (PAR4) antagonists based on a quinazolin-4(3H)-one scaffold.EBI
China Pharmaceutical University
Protease activated receptor 4 (PAR4) antagonists: Research progress on small molecules in the field of antiplatelet agents.EBI
China Pharmaceutical University
Development of a Series of (1-Benzyl-3-(6-methoxypyrimidin-3-yl)-5-(trifluoromethoxy)-1H-indol-2-yl)methanols as Selective Protease Activated Receptor 4 (PAR4) Antagonists with in Vivo Utility and Activity Against γ-Thrombin.EBI
Northwest Agriculture & Forestry University
Discovery of Potent Protease-Activated Receptor 4 Antagonists with in Vivo Antithrombotic Efficacy.EBI
Bristol-Myers Squibb Research & Development
Small Molecule Allosteric Modulators of G-Protein-Coupled Receptors: Drug-Target Interactions.EBI
Shanghai Jiao Tong University
Aliphatic prolinamide derivativesBDB
Orion Ophthalmology
Stereoselective inhibition of butyrylcholinesterase by enantiomers of exo- and endo-2-norbornyl-N-n-butylcarbamates.BDB
Chung Shan Medical University Hospital
Propellane-based compounds and the use thereofBDB
Purdue Pharma
Purinone derivative hydrochlorideBDB
Ono Pharmaceutical
Evaluation of 2-indolcarbohydrazones as potent a-glucosidase inhibitors, in silico studies and DFT based stereochemical predictions.BDB
Universiti Teknologi Mara (Uitm)
Substituted pyrrolidine-2-carboxamidesBDB
F. Hoffmann-La Roche