Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50006764
TargetProteinase-activated receptor 2(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50274114(CHEMBL4128763)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human PAR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50503155(CHEMBL4519152)
Affinity DataIC50: 170nMAssay Description:Negative allosteric modulation of CCR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProteinase-activated receptor 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50274114(CHEMBL4128763)
Affinity DataIC50: 380nMAssay Description:Antagonist activity at human PAR4More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50274114(CHEMBL4128763)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at human PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed