Compile Data Set for Download or QSAR
Report error Found 101 Enz. Inhib. hit(s) with all data for entry = 50014679
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578824(CHEMBL4860533)
Affinity DataIC50: 0.530nMAssay Description:Antagonist activity at human PAR4 expressed in Ga15-HEK293 cells assessed as reduction in PAR4 AP AYPGKF-NH2-induced cytosolic calcium incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM176061(US9688695, 94 | US10047103, 94)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human PAR4 expressed in Ga15-HEK293 cells assessed as reduction in PAR4 AP AYPGKF-NH2-induced cytosolic calcium incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578829(CHEMBL4855875)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human PAR4 expressed in Ga15-HEK293 cells assessed as reduction in PAR4 AP AYPGKF-NH2-induced cytosolic calcium incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578826(CHEMBL4871001)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human PAR4 expressed in Ga15-HEK293 cells assessed as reduction in PAR4 AP AYPGKF-NH2-induced cytosolic calcium incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM176003(US9688695, 36 | US10047103, 36)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578827(CHEMBL4866566)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human PAR4 expressed in Ga15-HEK293 cells assessed as reduction in PAR4 AP AYPGKF-NH2-induced cytosolic calcium incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578829(CHEMBL4855875)
Affinity DataIC50: 6.60nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578886(CHEMBL4849569)
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at human PAR4 expressed in Ga15-HEK293 cells assessed as reduction in PAR4 AP AYPGKF-NH2-induced cytosolic calcium incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM176061(US9688695, 94 | US10047103, 94)
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578824(CHEMBL4860533)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578827(CHEMBL4866566)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578886(CHEMBL4849569)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578826(CHEMBL4871001)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578824(CHEMBL4860533)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578828(CHEMBL4870185)
Affinity DataIC50: 107nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578827(CHEMBL4866566)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578886(CHEMBL4849569)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578829(CHEMBL4855875)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578825(CHEMBL4859532)
Affinity DataIC50: 174nMAssay Description:Antagonist activity at PAR4 in human platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turbidim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578875(CHEMBL4855377)
Affinity DataIC50: 520nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578828(CHEMBL4870185)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578820(CHEMBL4857938)
Affinity DataIC50: 790nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578826(CHEMBL4871001)
Affinity DataIC50: 830nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM364565(US9862730, Example 1 | 6-(Benzofuran-2-yl)-2-(meth...)
Affinity DataIC50: 940nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578878(CHEMBL4849478)
Affinity DataIC50: 950nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578823(CHEMBL4866983)
Affinity DataIC50: 980nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578850(CHEMBL4867779)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578824(CHEMBL4860533)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PAR2 expressed in Ga15-HEK293 cells assessed as reduction in PAR2 AP 2-furoyl-LIGRLO-NH2-induced cytosolic calcium incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM176061(US9688695, 94 | US10047103, 94)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PAR2 expressed in Ga15-HEK293 cells assessed as reduction in PAR2 AP 2-furoyl-LIGRLO-NH2-induced cytosolic calcium incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578826(CHEMBL4871001)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PAR2 expressed in Ga15-HEK293 cells assessed as reduction in PAR2 AP 2-furoyl-LIGRLO-NH2-induced cytosolic calcium incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578827(CHEMBL4866566)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PAR2 expressed in Ga15-HEK293 cells assessed as reduction in PAR2 AP 2-furoyl-LIGRLO-NH2-induced cytosolic calcium incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578886(CHEMBL4849569)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PAR2 expressed in Ga15-HEK293 cells assessed as reduction in PAR2 AP 2-furoyl-LIGRLO-NH2-induced cytosolic calcium incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578829(CHEMBL4855875)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human PAR2 expressed in Ga15-HEK293 cells assessed as reduction in PAR2 AP 2-furoyl-LIGRLO-NH2-induced cytosolic calcium incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578876(CHEMBL4871578)
Affinity DataIC50: 1.04E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578825(CHEMBL4859532)
Affinity DataIC50: 1.22E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578852(CHEMBL4867321)
Affinity DataIC50: 1.38E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578861(CHEMBL4849024)
Affinity DataIC50: 1.38E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578821(CHEMBL4871870)
Affinity DataIC50: 1.63E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM364589(US9862730, Example 41)
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578822(CHEMBL4847592)
Affinity DataIC50: 1.84E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578847(CHEMBL4858844)
Affinity DataIC50: 1.85E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578845(CHEMBL4860348)
Affinity DataIC50: 2.07E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578853(CHEMBL4864730)
Affinity DataIC50: 2.09E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578865(CHEMBL4865655)
Affinity DataIC50: 2.32E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578874(CHEMBL4859012)
Affinity DataIC50: 2.52E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578860(CHEMBL4862300)
Affinity DataIC50: 2.61E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578843(CHEMBL4855122)
Affinity DataIC50: 2.62E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578818(CHEMBL4848044)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578872(CHEMBL4849962)
Affinity DataIC50: 3.02E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteinase-activated receptor 4(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50578815(CHEMBL4855079)
Affinity DataIC50: 3.13E+3nMAssay Description:Antagonist activity at PAR4 in ICR mouse platelet-rich plasma assessed as inhibition of PAR4 AP AYPGKF-NH2-induced platelet aggregation by photo-turb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
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