22 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
Organization
Tritium-labelled isovaleryl-RYYRIK-NH2 as potential antagonist probe for ORL1 nociceptin receptor.
Kyushu University
20(S)-Ginsenoside Rh2 as aldose reductase inhibitor from Panax ginseng.
Kyushu University
Functional characterization of mouse cation transporter mOCT2 compared with mOCT1.
Kyushu University
Synthesis of 61-bis(1-adamantylcarbamoyl)-1,2-methano[60]fullerene and its antagonistic effect on haloperidol-induced catalepsy in mice.
Kyushu University
Spare interactions of highly potent [Arg(14),Lys(15)]nociceptin for cooperative induction of ORL1 receptor activation.
Kyushu University
Designed modification of partial agonist of ORL1 nociceptin receptor for conversion into highly potent antagonist.
Kyushu University
Differential receptor binding characteristics of consecutive phenylalanines in micro-opioid specific peptide ligand endomorphin-2.
Kyushu University
Discriminatory synergistic effect of Trp-substitutions in superagonist [(Arg/Lys)(14), (Arg/Lys)(15)]nociceptin on ORL1 receptor binding and activation.
Kyushu University
Discovery of Chlorofluoroacetamide-Based Covalent Inhibitors for Severe Acute Respiratory Syndrome Coronavirus 2 3CL Protease.
Kyushu University
Direct evidence of edge-to-face CH/π interaction for PAR-1 thrombin receptor activation.
Kyushu University
An electrochemical device for the assay of the interaction between a dioxin receptor and its various ligands.
Kyushu University
Solid-Phase synthesis of a library constructed of aromatic phosphate, long alkyl chains and tryptophane components, and identification of potent dipeptide telomerase inhibitors.
Kyushu University
Bisphenol AF: Halogen bonding effect is a major driving force for the dual ERα-agonist and ERβ-antagonist activities.
Kyushu University
Early identification of promiscuous attributes of aldose reductase inhibitors using a DMSO-perturbation assay.
Kyushu University
Design of new inhibitors for cdc2 kinase based on a multiple pseudosubstrate structure.
Kyushu University
Identification of the 5,5-dioxo-7,8-dihydro-6H-thiopyrano[3,2-d]pyrimidine derivatives as highly selective PDE4B inhibitors.
Kyushu University
Synthesis and biological evaluation of 5-carbamoyl-2-phenylpyrimidine derivatives as novel and potent PDE4 inhibitors.
Kyushu University
Ambuic acid inhibits the biosynthesis of cyclic peptide quormones in gram-positive bacteria.
Kyushu University
Design and synthesis of benzoacridines as estrogenic and anti-estrogenic agents.
Kyushu University
