Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50037943
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 1.13nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 1.89nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209307((S)-N-((S)-1-((S)-1-amino-1-oxo-3-(perfluorophenyl...)
Affinity DataIC50: 2.74nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataIC50: 3.46nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209302((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 11.7nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209304((S)-N-((S)-1-((S)-1-amino-1-oxohexan-2-ylamino)-1-...)
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209308((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50: 62nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209299((S)-N-((S)-1-((S)-1-amino-3-(4-hydroxyphenyl)-1-ox...)
Affinity DataIC50: 62.2nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209301(CHEMBL390914 | Morphiceptin [Val4] | (S)-1-((S)-2-...)
Affinity DataIC50: 76.5nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209300((S)-N-((S)-1-((S)-1-amino-1-oxopropan-2-ylamino)-1...)
Affinity DataIC50: 85.4nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50166048((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50: 87.1nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209314((S)-N-((S)-1-((S)-1-amino-3-(1H-imidazol-4-yl)-1-o...)
Affinity DataIC50: 138nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209298((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 148nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209316((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 230nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209311((S)-6-amino-5-((S)-2-((S)-1-((S)-2-amino-3-(4-hydr...)
Affinity DataIC50: 408nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 727nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209305((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50: 917nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209309((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 926nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209315((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209303((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 2.65E+3nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209298((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 3.15E+3nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 3.58E+3nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209313(H-Tyr-Pro-Ala-Phe-NH2 | YPAF-NH2 | (S)-N-((S)-1-((...)
Affinity DataIC50: 3.81E+3nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209306((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 4.49E+3nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209315((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 5.72E+3nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209307((S)-N-((S)-1-((S)-1-amino-1-oxo-3-(perfluorophenyl...)
Affinity DataIC50: 8.04E+3nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataIC50: 1.03E+4nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209305((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50: 1.14E+4nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209302((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.17E+4nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209316((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.52E+4nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209299((S)-N-((S)-1-((S)-1-amino-3-(4-hydroxyphenyl)-1-ox...)
Affinity DataIC50: 5.45E+4nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209304((S)-N-((S)-1-((S)-1-amino-1-oxohexan-2-ylamino)-1-...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209303((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209314((S)-N-((S)-1-((S)-1-amino-3-(1H-imidazol-4-yl)-1-o...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209301(CHEMBL390914 | Morphiceptin [Val4] | (S)-1-((S)-2-...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50166048((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209306((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209309((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209308((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50209310((S)-6-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [3H]DAGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed