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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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13 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Thienopyrimidines asß3-adrenoceptor agonists: hit-to-lead optimization.EBI
4Sc
A vHTS approach for the identification of beta-adrenoceptor ligands.EBI
4Sc
Substituted 2-arylbenzothiazoles as kinase inhibitors: hit-to-lead optimization.EBI
4Sc
Inhibitors of potassium channels KV1.3 and IK-1 as immunosuppressants.EBI
4Sc
N-substituted 2'-(aminoaryl)benzothiazoles as kinase inhibitors: hit identification and scaffold hopping.EBI
4Sc
Discovery of 5-HT6 receptor ligands based on virtual HTS.EBI
4Sc
SAR, species specificity, and cellular activity of cyclopentene dicarboxylic acid amides as DHODH inhibitors.EBI
4Sc
Discovery of a novel series of DHODH inhibitors by a docking procedure and QSAR refinement.EBI
4Sc
Heterocyclic compounds and uses thereofBDB
Nuvation Bio
Compounds IBDB
Benevolentai Cambridge
Necrosis inhibitorsBDB
National Institute of Biological Sciences, Beijing
Kinase inhibitorsBDB
Respivert
N-(cycloalkylamino)acyl-2-aminothiazole inhibitors of cyclin-dependent kinase 2. N-[5-[[[5-(1,1-dimethylethyl)-2-oxazolyl]methyl]thio]-2-thiazolyl]-4- piperidinecarboxamide (BMS-387032), a highly efficacious and selective antitumor agent.BDB
Bristol-Myers Squibb