Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50028427
LigandPNGBDBM50279106(5-(4-phenoxybutoxy)psoralen | 4-(4-phenoxybutoxy)-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)
Affinity DataIC50: 20nMAssay Description:Inhibition of IK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM31774(cid_2812 | CHEMBL104 | Canesten | Mycelex | Lotrim...)
Affinity DataIC50: 70nMAssay Description:Inhibition of IK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM31774(cid_2812 | CHEMBL104 | Canesten | Mycelex | Lotrim...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279024((1,3-dimethyl-1H-pyrazol-5-yl)(5-(furan-2-carbonyl...)
Affinity DataIC50: 710nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278971(2-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279105(5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278972(methyl 2-(5-(furan-2-carbonyl)-5,6-dihydrophenanth...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279065(5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278973((5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6-y...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278994(phenanthridine-5,6(6H)-diylbis(furan-2-ylmethanone...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278938(1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279063(5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one | CHEMBL49...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279105(5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279066(5-(3-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279104(5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278939((6-(cyclobutanecarbonyl)phenanthridin-5(6H)-yl)(fu...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278936(1-(6-(1H-indol-3-yl)phenanthridin-5(6H)-yl)ethanon...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279063(5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one | CHEMBL49...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM31774(cid_2812 | CHEMBL104 | Canesten | Mycelex | Lotrim...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279065(5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278937(1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279106(5-(4-phenoxybutoxy)psoralen | 4-(4-phenoxybutoxy)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279064(5-(4-nitrophenylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of cloned Kv1.3 channel expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279104(5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed