Compile Data Set for Download or QSAR
Report error Found 320 Enz. Inhib. hit(s) with all data for entry = 50028244
TargetEpidermal growth factor receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM4626(CHEMBL301018 | N-(3-chloro-4-fluorophenyl)-6,7-dim...)
Affinity DataIC50: 1nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM4626(CHEMBL301018 | N-(3-chloro-4-fluorophenyl)-6,7-dim...)
Affinity DataIC50: 24nMAssay Description:Inhibition of ErbB2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248349(N-(4-(benzo[d]thiazol-2-yl)-3-methoxyphenyl)-6,7-d...)
Affinity DataIC50: 63nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248413(N2-(3-(benzo[d]thiazol-2-yl)phenyl)-N4-(5-methyl-1...)
Affinity DataIC50: 100nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248293(N-(4-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxyqu...)
Affinity DataIC50: 135nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248413(N2-(3-(benzo[d]thiazol-2-yl)phenyl)-N4-(5-methyl-1...)
Affinity DataIC50: 160nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248413(N2-(3-(benzo[d]thiazol-2-yl)phenyl)-N4-(5-methyl-1...)
Affinity DataIC50: 190nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 190nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248294(N-(4-(benzo[d]thiazol-2-yl)-2-methylphenyl)-6,7-di...)
Affinity DataIC50: 240nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 280nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248229(N-(4-(benzo[d]thiazol-2-yl)-2-fluorophenyl)thieno[...)
Affinity DataIC50: 290nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248292(N-(4-(benzo[d]thiazol-2-yl)phenyl)-7-chloro-6-meth...)
Affinity DataIC50: 300nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 310nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248147(N2-(4-(benzo[d]thiazol-2-yl)-3-methoxyphenyl)-N4-(...)
Affinity DataIC50: 320nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248293(N-(4-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxyqu...)
Affinity DataIC50: 350nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248146(N2-(4-(benzo[d]thiazol-2-yl)phenyl)-N4-(5-methyl-1...)
Affinity DataIC50: 370nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM4626(CHEMBL301018 | N-(3-chloro-4-fluorophenyl)-6,7-dim...)
Affinity DataIC50: 480nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248232(N-(4-(benzo[d]thiazol-2-yl)-3-chlorophenyl)-7-chlo...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(N-(4-(benzo[d]thiazol-2-yl)-2-fluorophenyl)-7-chlo...)
Affinity DataIC50: 510nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM4626(CHEMBL301018 | N-(3-chloro-4-fluorophenyl)-6,7-dim...)
Affinity DataIC50: 510nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248232(N-(4-(benzo[d]thiazol-2-yl)-3-chlorophenyl)-7-chlo...)
Affinity DataIC50: 600nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 610nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248350(N4-(4-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxy-...)
Affinity DataIC50: 630nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248230(N-(4-(benzo[d]thiazol-2-yl)phenyl)-7-chloroquinoli...)
Affinity DataIC50: 630nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248230(N-(4-(benzo[d]thiazol-2-yl)phenyl)-7-chloroquinoli...)
Affinity DataIC50: 640nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248291(N-(4-(benzo[d]thiazol-2-yl)-2-fluorophenyl)-7-chlo...)
Affinity DataIC50: 700nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248185(N-(4-(benzo[d]thiazol-2-yl)phenyl)thieno[3,2-d]pyr...)
Affinity DataIC50: 720nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248149(N-(4-(benzo[d]thiazol-2-yl)-3-methoxyphenyl)-7H-py...)
Affinity DataIC50: 720nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248230(N-(4-(benzo[d]thiazol-2-yl)phenyl)-7-chloroquinoli...)
Affinity DataIC50: 750nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248414(N4-(3-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxy-...)
Affinity DataIC50: 780nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(N-(4-(benzo[d]thiazol-2-yl)-3-chlorophenyl)-7-chlo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248291(N-(4-(benzo[d]thiazol-2-yl)-2-fluorophenyl)-7-chlo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248232(N-(4-(benzo[d]thiazol-2-yl)-3-chlorophenyl)-7-chlo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248232(N-(4-(benzo[d]thiazol-2-yl)-3-chlorophenyl)-7-chlo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248414(N4-(3-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxy-...)
Affinity DataIC50: 810nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248120(N-(4-(benzo[d]thiazol-2-yl)phenyl)-4-(4-methylpipe...)
Affinity DataIC50: 840nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248416(N-(3-(benzo[d]thiazol-2-yl)phenyl)-9H-purin-6-amin...)
Affinity DataIC50: 840nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248294(N-(4-(benzo[d]thiazol-2-yl)-2-methylphenyl)-6,7-di...)
Affinity DataIC50: 840nMAssay Description:Inhibition of TIE2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248230(N-(4-(benzo[d]thiazol-2-yl)phenyl)-7-chloroquinoli...)
Affinity DataIC50: 860nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248416(N-(3-(benzo[d]thiazol-2-yl)phenyl)-9H-purin-6-amin...)
Affinity DataIC50: 870nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 900nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 900nMAssay Description:Inhibition of FAK by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248464(N-[4-(isoindolin-2-yl)phenyl]-6',7'-dimethoxyquina...)
Affinity DataIC50: 920nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248414(N4-(3-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxy-...)
Affinity DataIC50: 940nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248414(N4-(3-(benzo[d]thiazol-2-yl)phenyl)-6,7-dimethoxy-...)
Affinity DataIC50: 960nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248182(N-(4-(benzo[d]thiazol-2-yl)-3-methoxyphenyl)-2-met...)
Affinity DataIC50: 960nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50248085(N-(3-(benzo[d]thiazol-2-yl)-4-hydroxyphenylcarbamo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of VEGFR3 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(N-(4-(benzo[d]thiazol-2-yl)-2-fluorophenyl)-7-chlo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EphB4 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
4Sc

Curated by ChEMBL
LigandPNGBDBM50248291(N-(4-(benzo[d]thiazol-2-yl)-2-fluorophenyl)-7-chlo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TIE2 by virtual HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Displayed 1 to 50 (of 320 total ) | Next | Last >>
Jump to: