Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.
Human
Ki: 1
Calcium release-activated calcium channel protein 1/Short transient receptor potential channel 1/Short transient receptor potential channel 3/Stromal interaction molecule 1 P48995 Q13507 Q13586 Q96D31
Human
IC50: 1
Human
IC50: 15
Human
CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II SUBUNIT ALPHA P08413 P11275 Q13554 Q13555 Q13557 Q9UQM7
Rat
Human
Rat
EC50: 1
CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II SUBUNIT BETA P08413 P11275 Q13554 Q13555 Q13557 Q9UQM7
Rat
EC50: 1
Calcium/calmodulin-dependent protein kinase type II subunit alpha/beta/delta/gamma Q13554 Q13555 Q13557 Q9UQM7
Human
IC50: 26
Human
CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II SUBUNIT DELTA P11730 P15791 Q13554 Q13555 Q13557 Q9UQM7
Calcium/calmodulin-dependent protein kinase type II subunit alpha/beta/delta/gamma Q13554 Q13555 Q13557 Q9UQM7
Human
IC50: 26
Human
CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II SUBUNIT GAMMA P11730 P15791 Q13554 Q13555 Q13557 Q9UQM7
Calcium/calmodulin-dependent protein kinase type II subunit alpha/beta/delta/gamma Q13554 Q13555 Q13557 Q9UQM7
Human
IC50: 26
Rat
EC50: 1
Human
Human
CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT ALPHA O95067 P00517 P05132 P06493 P14635 P17612 P22612 P22694 P27791 Q8WWL7 Q95J97
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3/cAMP-dependent protein kinase O95067 P06493 P14635 Q8WWL7 Q95J97
Rabbit
IC50: 1
Mouse
Human
Bovine
IC50: 5
Bovine
IC50: 1
Bovine
IC50: 5
Bovine
IC50: 5
Bovine
IC50: 5
Bovine
IC50: 5
Bovine
IC50: 3
Human
Human
Human
CANNABINOID RECEPTOR 1 A0A0H4AWC7 A0A0V1DID4 P20272 P21554 P34972 P47746 P47936 P56971 Q17QM9 Q99NU1 Q9PUI7 Q9QZN9
Human
CARBONIC ANHYDRASE A0A086SLX8 A0A952HKT9 A6YCJ1 B5SU02 C0IX24 O24855 P40881 P46510 P53615 P96878 Q08IJ2 Q2PCB5 Q3I4V7 Q50565 Q5AJ71 Q5TU56 Q6FTL6 Q9HVB9 Q9KMP6 Q9V396 Q9ZK30 R4ML78
Ki: 1283
Helicobacter pylori (strain J99 / ATCC 700824) (Campylobacter pylori J99)
Ki: 47
Cryptococcus neoformans var. grubii (Filobasidiella neoformans var. grubii)
Ki: 93
Vibrio cholerae serotype O1 (strain ATCC 39315 / El Tor Inaba N16961)
Ki: 37
Helicobacter pylori (strain ATCC 700392 / 26695) (Campylobacterpylori)
Ki: 35
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Ki: 107
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228)
Ki: 37
CARBONIC ANHYDRASE 1 O43570 P00915 P00916 P00917 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 12 O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
Human
CARBONIC ANHYDRASE 13 O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9D6N1 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 14 O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
Human
CARBONIC ANHYDRASE 2 O43570 P00915 P00918 P00921 P07451 P18915 P22748 P23280 P27139 P35218 P43166 P9WPJ9 Q16790 Q3SZX4 Q8N1Q1 Q95323 Q9ULX7 Q9Y2D0
Carbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9 O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
Human
Human
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Ki: 66
CARBONIC ANHYDRASE 3 O43570 P00915 P00918 P00921 P07451 P18915 P22748 P23280 P35218 P43166 Q16790 Q3SZX4 Q8N1Q1 Q95323 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 4 O43570 P00915 P00918 P00921 P07451 P18915 P22748 P23280 P35218 P43166 Q16790 Q3SZX4 Q8N1Q1 Q95323 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 5A, MITOCHONDRIAL O43570 P00915 P00918 P07451 P22748 P23280 P23589 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 5B, MITOCHONDRIAL O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
Human
CARBONIC ANHYDRASE 6 O43570 P00915 P00918 P00921 P07451 P18915 P22748 P23280 P35218 P43166 Q16790 Q3SZX4 Q8N1Q1 Q95323 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 7 O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ERQ8 Q9ULX7 Q9Y2D0
CARBONIC ANHYDRASE 9 O43570 P00915 P00918 P07451 P22748 P23280 P35218 P43166 Q16790 Q8N1Q1 Q9ULX7 Q9Y2D0
Human
Porphyromonas gingivalis (Bacteroides gingivalis)
Ki: 4
Human
IC50: 9
Human
IC50: 9
Human
IC50: 9
Human
IC50: 9
Human
IC50: 1
Human
Human
IC50: 1
Human
Human
Human
CASPASE-3 P29466 P31944 P42574 P42575 P49662 P51878 P55210 P55211 P55212 P70677 Q14790 Q6UXS9 Q92851
CASPASE-4 P29466 P31944 P42574 P42575 P49662 P51878 P55210 P55211 P55212 P70343 Q14790 Q6UXS9 Q92851
Human
Human
Human
Human
Human
Human
Ki: 7
Human
Human
Human
Human
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228)
IC50: 9
Human
Human
Human
Human
Human
CGMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE O54735 O76074 O77746 P51160 P54750 Q01064 Q14123 Q28156
Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha'/cGMP-specific 3',5'-cyclic phosphodiesterase O76074 P51160
Human
Ki: 4
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A/1B/1C/cGMP-specific 3',5'-cyclic phosphodiesterase O76074 P54750 Q01064 Q14123
Human
IC50: 51
Human
Human
IC50: 3
Human
IC50: 165
Human
IC50: 165
Human
IC50: 165
Mitochondrial complex I (NADH dehydrogenase) O00217 O00483 O14561 O15239 O43181 O43674 O43676 O43677 O43678 O43920 O75251 O75306 O75380 O75438 O75489 O95139 O95167 O95168 O95169 O95178 O95182 O95298 O95299 O96000 P03886 P03891 P03897 P03901 P03905 P03915 P03923 P17568 P19404 P28331 P49821 P51970 P56181 P56556 Q16718 Q16795 Q86Y39 Q8N183 Q9BU61 Q9NRX3 Q9NX14 Q9P032 Q9P0J0 Q9UI09 Q9Y375 Q9Y6M9
Human
IC50: 1
CONE CGMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE SUBUNIT ALPHA' O43924 O76074 P04972 P11541 P16499 P16586 P18545 P22571 P23439 P35913 P51160 Q13956 Q95142
Human
Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha'/cGMP-specific 3',5'-cyclic phosphodiesterase O76074 P51160
Human
Ki: 4
Human
Human
Human
CYCLIN-DEPENDENT KINASE 1 O95067 P00546 P06493 P11440 P14635 P15206 P20248 P24864 P30281 Q8WWL7 Q95J97 Q9DGD3
Spiny starfish
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3 O95067 P06493 P14635 Q8WWL7
Human
CYCLIN-DEPENDENT KINASE 2 O96020 P09211 P20248 P22674 P24385 P24864 P24941 P30274 P30279 P78396 Q8ND76
Human
Human
Human
IC50: 2
Human
IC50: 2
Human
Human
Human
Human
IC50: 41
Human
Human
Human
Cryptosporidium parvum (strain Iowa II)
IC50: 1
Human
Human
Mouse
Human
Human
Human
Human
Human
CYTOCHROME C OXIDASE SUBUNIT NDUFA4 O00217 O00483 O14561 O15239 O43181 O43674 O43676 O43677 O43678 O43920 O75251 O75306 O75380 O75438 O75489 O95139 O95167 O95168 O95169 O95178 O95182 O95298 O95299 O96000 P03886 P03891 P03897 P03901 P03905 P03915 P03923 P17568 P19404 P28331 P49821 P51970 P56181 P56556 Q16718 Q16795 Q86Y39 Q8N183 Q9BU61 Q9NRX3 Q9NX14 Q9P032 Q9P0J0 Q9UI09 Q9Y375 Q9Y6M9
Human
IC50: 5
Mitochondrial complex I (NADH dehydrogenase) O00217 O00483 O14561 O15239 O43181 O43674 O43676 O43677 O43678 O43920 O75251 O75306 O75380 O75438 O75489 O95139 O95167 O95168 O95169 O95178 O95182 O95298 O95299 O96000 P03886 P03891 P03897 P03901 P03905 P03915 P03923 P17568 P19404 P28331 P49821 P51970 P56181 P56556 Q16718 Q16795 Q86Y39 Q8N183 Q9BU61 Q9NRX3 Q9NX14 Q9P032 Q9P0J0 Q9UI09 Q9Y375 Q9Y6M9
Human
IC50: 1
Mycobacterium tuberculosis (strain CDC 1551 / Oshkosh)
Kd: 7
Mycobacterium tuberculosis (strain CDC 1551 / Oshkosh)
Kd: 6
CYTOCHROME P450 1A1 P00185 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 1A2 P00186 P04798 P04799 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 1B1 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2A13 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2A6 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2B6 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2C18 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2C19 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2C8 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2C9 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2D6 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2E1 P04798 P05177 P05181 P05182 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 2J2 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 3A4 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 3A43 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 3A5 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 3A7 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 4A11 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 4B1 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 4F2 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 4F3 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55
CYTOCHROME P450 4F8 P04798 P05177 P05181 P08684 P10632 P10635 P11509 P11712 P13584 P20813 P20815 P20853 P24462 P24903 P33260 P33261 P51589 P78329 P98187 Q02928 Q08477 Q16678 Q16696 Q5TCH4 Q6VVX0 Q746J6 Q7Z449 Q8TAV3 Q96SQ9 Q9HB55

