BindingDB

The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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To help with training and testing AI and other models, BindingDB downloads and search results now provide the publication date and BindingDB curation date of each measurement.

18 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Revisiting 1,3,4-Oxadiazol-2-ones: Utilization in the Development of ABHD6 Inhibitors.EBI
University of Eastern Finland
Piperazine and piperidine carboxamides and carbamates as inhibitors of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL).EBI
University of Eastern Finland
Loratadine analogues as MAGL inhibitors.EBI
University of Eastern Finland
Rational design of novel CYP2A6 inhibitors.EBI
University of Eastern Finland
Discovery of 5-benzyl-3-phenyl-4,5-dihydroisoxazoles and 5-benzyl-3-phenyl-1,4,2-dioxazoles as potent firefly luciferase inhibitors.EBI
University of Eastern Finland
Chiral 1,3,4-oxadiazol-2-ones as highly selective FAAH inhibitors.EBI
University of Eastern Finland
Screen of pseudopeptidic inhibitors of human sirtuins 1-3: two lead compounds with antiproliferative effects in cancer cells.EBI
University of Eastern Finland
The use of novel C-methylated spermidine derivatives to investigate the regulation of polyamine metabolism.EBI
University of Eastern Finland
Design, synthesis, and biological evaluation of nonsteroidal cycloalkane[d]isoxazole-containing androgen receptor modulators.EBI
University of Eastern Finland
Antifungal activities of novel non-azole molecules against S. cerevisiae and C. albicans.EBI
University of Eastern Finland
Identification of novel CYP2A6 inhibitors by virtual screening.EBI
University of Eastern Finland
Structure-based design of pseudopeptidic inhibitors for SIRT1 and SIRT2.EBI
University of Eastern Finland
N(epsilon)-Modified lysine containing inhibitors for SIRT1 and SIRT2.EBI
University of Eastern Finland
Design, synthesis and in vitro/in vivo evaluation of orally bioavailable prodrugs of a catechol-O-methyltransferase inhibitor.EBI
University of Eastern Finland
A Selective and Slowly Reversible Inhibitor of l-Type Amino Acid Transporter 1 (LAT1) Potentiates Antiproliferative Drug Efficacy in Cancer Cells.EBI
University of Eastern Finland
Potent and selective N-(4-sulfamoylphenyl)thiourea-based GPR55 agonists.EBI
University of Eastern Finland
Microwave-assisted synthesis of quinoline, isoquinoline, quinoxaline and quinazoline derivatives as CB2 receptor agonists.EBI
University of Eastern Finland
Augmentation of Anticancer Drug Efficacy in Murine Hepatocellular Carcinoma Cells by a Peripherally Acting Competitive N-Methyl-d-aspartate (NMDA) Receptor Antagonist.EBI
University of Eastern Finland