Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50040411
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM8885(Testosterone, 1 | (1S,2R,10R,11S,14S,15S)-14-hydro...)
Affinity DataIC50: 4.57nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393821(CHEMBL2159566)
Affinity DataIC50: 27.5nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393813(CHEMBL2159561)
Affinity DataIC50: 43.6nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393819(CHEMBL2159568)
Affinity DataIC50: 64.6nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393819(CHEMBL2159568)
Affinity DataIC50: 64.6nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393810(CHEMBL2159540)
Affinity DataIC50: 105nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM18678(CHEMBL63560 | (2R)-N-[4-cyano-3-(trifluoromethyl)p...)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393818(CHEMBL2159569)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393817(CHEMBL2159570)
Affinity DataIC50: 129nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393828(CHEMBL2159730)
Affinity DataIC50: 224nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM35909(Eulexin | 2-hydroxy-2-methyl-N-(4-nitro-3-(trifluo...)
Affinity DataIC50: 224nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393816(CHEMBL2159571)
Affinity DataIC50: 263nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393824(CHEMBL2159563)
Affinity DataIC50: 269nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393805(CHEMBL2159545)
Affinity DataIC50: 295nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393825(CHEMBL2159562)
Affinity DataIC50: 302nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393809(CHEMBL2159541)
Affinity DataIC50: 309nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393808(CHEMBL2159542)
Affinity DataIC50: 389nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393827(CHEMBL2159731)
Affinity DataIC50: 447nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393829(CHEMBL2159729)
Affinity DataIC50: 617nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393806(CHEMBL2159544)
Affinity DataIC50: 660nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393806(CHEMBL2159544)
Affinity DataIC50: 661nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393803(CHEMBL2159547)
Affinity DataIC50: 708nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393802(CHEMBL2159548)
Affinity DataIC50: 741nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393802(CHEMBL2159548)
Affinity DataIC50: 776nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393814(CHEMBL2159573)
Affinity DataIC50: 977nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393814(CHEMBL2159573)
Affinity DataIC50: 977nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393811(CHEMBL2159539)
Affinity DataIC50: 999nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393811(CHEMBL2159539)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393815(CHEMBL2159572)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393820(CHEMBL2159567)
Affinity DataIC50: 1.14E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393820(CHEMBL2159567)
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393823(CHEMBL2159564)
Affinity DataIC50: 1.48E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393822(CHEMBL2159565)
Affinity DataIC50: 1.54E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393822(CHEMBL2159565)
Affinity DataIC50: 1.55E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393804(CHEMBL2159546)
Affinity DataIC50: 1.99E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393804(CHEMBL2159546)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393826(CHEMBL2159732)
Affinity DataIC50: 2.51E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393801(CHEMBL2159549)
Affinity DataIC50: 2.81E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393801(CHEMBL2159549)
Affinity DataIC50: 2.82E+3nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393807(CHEMBL2159543)
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50393812(CHEMBL2159550)
Affinity DataIC50: 1.32E+4nMAssay Description:Displacement of [3H]R1881 from wild type human androgen receptor expressed in COS-1 cells co-transfected with pSG5 after 15 mins by scintillation ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed