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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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11 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of novel furanone derivatives as potent Cdc7 kinase inhibitors.EBI
Carna Biosciences
TR-FRET binding assay targeting unactivated form of Bruton's tyrosine kinase.EBI
Carna Biosciences
Design and combinatorial synthesis of a novel kinase-focused library using click chemistry-based fragment assembly.EBI
Carna Biosciences
Discovery of AS-1763: A Potent, Selective, Noncovalent, and Orally Available Inhibitor of Bruton's Tyrosine Kinase.EBI
Carna Biosciences
Discovery of AS-0141, a Potent and Selective Inhibitor of CDC7 Kinase for the Treatment of Solid Cancers.EBI
Carna Biosciences
Identification of an allosteric and Smad3-selective inhibitor of p38αMAPK using a substrate-based approach.EBI
Carna Biosciences
Design and Synthesis of Novel Amino-triazine Analogues as Selective Bruton's Tyrosine Kinase Inhibitors for Treatment of Rheumatoid Arthritis.EBI
Carna Biosciences
Design and synthesis of novel pyrimidine analogs as highly selective, non-covalent BTK inhibitors.EBI
Carna Biosciences
Bicyclic compounds as ATX inhibitorsBDB
Hoffmann-La Roche
Derivatives of 6-(2,3-dichlorophenyl)-1,2,4-triazin-5-amineBDB
Nektar Therapeutics
2-styrylchromones as novel inhibitors of xanthine oxidase. A structure-activity study.BDB
University of Porto-Rua Anibal Cunha