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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of SENP1 inhibitors through in silico screening and rational drug design.EBI
Shanghai Jiao Tong University
Development and evaluation of a highly reliable assay for SUMO-specific protease inhibitors.EBI
Shanghai Jiao Tong University
Spongiacidin C, a pyrrole alkaloid from the marine sponge Stylissa massa, functions as a USP7 inhibitor.EBI
Kumamoto University
Discovery of 1-[4-(N-benzylamino)phenyl]-3-phenylurea derivatives as non-peptidic selective SUMO-sentrin specific protease (SENP)1 inhibitors.EBI
Gakushuin University
2-(4-Chlorophenyl)-2-oxoethyl 4-benzamidobenzoate derivatives, a novel class of SENP1 inhibitors: Virtual screening, synthesis and biological evaluation.EBI
Shanghai Jiao Tong University
Design, synthesis, and biological evaluation of benzodiazepine-based SUMO-specific protease 1 inhibitors.EBI
Shanghai Jiao Tong University
Recent research and development of inhibitors targeting sentrin-specific protease 1 for the treatment of cancers.EBI
Sichuan University
Discovery and radiosensitization research of ursolic acid derivatives as SENP1 inhibitors.EBI
Peking Union Medical College
Discovery of Natural Ursane-type SENP1 Inhibitors and the Platinum Resistance Reversal Activity Against Human Ovarian Cancer Cells: A Structure-Activity Relationship Study.EBI
Peking Union Medical College
Small-molecule inhibitors targeting small ubiquitin-like modifier pathway for the treatment of cancers and other diseases.EBI
China Pharmaceutical University
Benzothiophene-2-carboxamide derivatives as SENPs inhibitors with selectivity within SENPs family.EBI
Shanghai Jiao Tong University
Vialinin A and thelephantin G, potent inhibitors of tumor necrosis factor-α production, inhibit sentrin/SUMO-specific protease 1 enzymatic activity.EBI
Tokyo University of Agriculture
Apoptosis signal-regulating kinase inhibitors and uses thereofBDB
Sichuan Haisco Pharmaceutical
Synthesis, in vitro evaluation and molecular docking studies of novel coumarin-isatin derivatives as a-glucosidase inhibitors.BDB
Jishou University
Potent cationic inhibitors of West Nile virus NS2B/NS3 protease with serum stability, cell permeability and antiviral activity.BDB
University of Queensland