Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50040456
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394464(CHEMBL2159857)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394465(CHEMBL2159858)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394468(CHEMBL2159859)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394466(CHEMBL2159862)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394467(CHEMBL2159861)
Affinity DataIC50: 2.39E+3nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394469(CHEMBL2159860)
Affinity DataIC50: 3.54E+3nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394460(CHEMBL2159852)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394461(CHEMBL2159854)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394462(CHEMBL2159856)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSentrin-specific protease 1(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50394463(CHEMBL2159855)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant His-tagged SENP1 catalytic domain expressed in Escherichia coli BL21(DE3) using His-tagged deltaRanGAP-SUMO2 as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed