BindingDB

The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.5M data for 728K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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15 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of N-(2-oxoethyl) sulfanilamide-derived inhibitors of KAT6A (MOZ) against leukemia by an isostere strategy.EBI
Children's Hospital Affiliated to Zhengzhou University
Acetyl-Click Screening Platform Identifies Small-Molecule Inhibitors of Histone Acetyltransferase 1 (HAT1).EBI
Wayne State University
First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8.EBI
Sapienza University of Rome
Discovery of DS-9300: A Highly Potent, Selective, and Once-Daily Oral EP300/CBP Histone Acetyltransferase Inhibitor.EBI
Daiichi Sankyo Co.
Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring.EBI
Daiichi Sankyo
4-Pyridone-3-carboxylic acid as a benzoic acid bioisostere: Design, synthesis, and evaluation of EP300/CBP histone acetyltransferase inhibitors.EBI
Daiichi Sankyo
Histone acetyltransferase inhibitors: An overview in synthesis, structure-activity relationship and molecular mechanism.EBI
Sichuan University
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A.EBI
Cancer Therapeutics Crc
ANTIBIOTIC PYRAZINOTHIAZINE DERIVATIVES AND PROCESS OF PREPARATION THEREOFBDB
Bugworks Research India
FUNCTIONALIZED AMINOTHIAZOLESBDB
Leadxpro
Substituted heterocycles as aldehyde dehydrogenase inhibitorsBDB
Kayothera
Mu opioid receptor modulatorsBDB
University of California
2,3-dihydrofuro[2,3-b]pyridine compoundsBDB
Eli Lilly
Selective inhibitors of protein arginine methyltransferase 5 (PRMT5)BDB
Prelude Therapeutics
Methylamine derivatives as lysysl oxidase inhibitors for the treatment of cancerBDB
The Institute of Cancer Research: Royal Cancer Hospital