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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis of dihydroimidazole tethered imidazolinethiones and their activity as novel antagonists of the nuclear retinoic acid receptor-related orphan receptors (RORs).EBI
Torrey Pines Institute For Molecular Studies
Potentµ-Opioid Receptor Agonists from Cyclic Peptides Tyr-c[D-Lys-Xxx-Tyr-Gly]: Synthesis, Biological, and Structural Evaluation.EBI
Torrey Pines Institute For Molecular Studies
Parallel Synthesis of Hexahydrodiimidazodiazepines Heterocyclic Peptidomimetics and Their in Vitro and in Vivo Activities atµ (MOR),d (DOR), and¿ (KOR) Opioid Receptors.EBI
Torrey Pines Institute For Molecular Studies
Discovery of a potent and selectivea3ß4 nicotinic acetylcholine receptor antagonist from ana-conotoxin synthetic combinatorial library.EBI
Torrey Pines Institute For Molecular Studies
Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies.EBI
Torrey Pines Institute For Molecular Studies
Furin inhibitors: importance of the positive formal charge and beyond.EBI
Torrey Pines Institute For Molecular Studies
Recent advances in the synthesis of raloxifene: a selective estrogen receptor modulator.EBI
Torrey Pines Institute For Molecular Studies
Conformation-opioid activity relationships of bicyclic guanidines from 3D similarity analysis.EBI
Torrey Pines Institute For Molecular Studies
Mixture-based synthetic combinatorial libraries.EBI
Torrey Pines Institute For Molecular Studies
Discovery of a novel protein kinase B inhibitor by structure-based virtual screening.EBI
Torrey Pines Institute For Molecular Studies
Highly Selective and Potentα4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats.EBI
Torrey Pines Institute For Molecular Studies
Pyridine derivativesBDB
Hoffmann-La Roche