Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50039714
TargetEstrogen receptor(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382735(CHEMBL2024377)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161712((4-Chloro-phenyl)-(4-{4-[6-hydroxy-2-(4-hydroxy-ph...)
Affinity DataIC50: 0.220nMAssay Description:Displacement of [3H]-17beta-estradiol from ERalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161706((4-{4-[6-Hydroxy-2-(4-hydroxy-phenyl)-benzo[b]thio...)
Affinity DataIC50: 0.270nMAssay Description:Displacement of [3H]-17beta-estradiol from ERalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161698([6-Hydroxy-2-(4-hydroxy-phenyl)-benzo[b]thiophen-3...)
Affinity DataIC50: 0.280nMAssay Description:Displacement of [3H]-17beta-estradiol from ERalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382734(CHEMBL2024376)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382735(CHEMBL2024377)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382734(CHEMBL2024376)
Affinity DataIC50: 3.10nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161712((4-Chloro-phenyl)-(4-{4-[6-hydroxy-2-(4-hydroxy-ph...)
Affinity DataIC50: 9.07nMAssay Description:Displacement of [3H]-17beta-estradiol from ERbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161706((4-{4-[6-Hydroxy-2-(4-hydroxy-phenyl)-benzo[b]thio...)
Affinity DataIC50: 12.5nMAssay Description:Displacement of [3H]-17beta-estradiol from ERbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161698([6-Hydroxy-2-(4-hydroxy-phenyl)-benzo[b]thiophen-3...)
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]-17beta-estradiol from ERbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed