Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50049171
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235609(CHEMBL4096280)
Affinity DataIC50: 5.10E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235608(CHEMBL4067306)
Affinity DataIC50: 5.60E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235602(CHEMBL4101440)
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235604(CHEMBL4088559)
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235608(CHEMBL4067306)
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235621(CHEMBL4071074)
Affinity DataIC50: 6.30E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235607(CHEMBL4091903)
Affinity DataIC50: 6.30E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235602(CHEMBL4101440)
Affinity DataIC50: 6.40E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235609(CHEMBL4096280)
Affinity DataIC50: 6.40E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235617(CHEMBL4083451)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235620(CHEMBL4063381)
Affinity DataIC50: 6.60E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235607(CHEMBL4091903)
Affinity DataIC50: 6.80E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235620(CHEMBL4063381)
Affinity DataIC50: 6.80E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235617(CHEMBL4083451)
Affinity DataIC50: 7.50E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235603(CHEMBL4091239)
Affinity DataIC50: 7.70E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235622(CHEMBL4085975)
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235621(CHEMBL4071074)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235609(CHEMBL4096280)
Affinity DataIC50: 8.30E+3nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235622(CHEMBL4085975)
Affinity DataIC50: 8.40E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235621(CHEMBL4071074)
Affinity DataIC50: 8.40E+3nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235607(CHEMBL4091903)
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235608(CHEMBL4067306)
Affinity DataIC50: 9.10E+3nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235623(CHEMBL4064439)
Affinity DataIC50: 9.30E+3nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235603(CHEMBL4091239)
Affinity DataIC50: 9.90E+3nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235619(CHEMBL4073023)
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235602(CHEMBL4101440)
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235618(CHEMBL4093723)
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235622(CHEMBL4085975)
Affinity DataIC50: 1.07E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235617(CHEMBL4083451)
Affinity DataIC50: 1.09E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235606(CHEMBL4067157)
Affinity DataIC50: 1.18E+4nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235618(CHEMBL4093723)
Affinity DataIC50: 1.19E+4nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235620(CHEMBL4063381)
Affinity DataIC50: 1.24E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235603(CHEMBL4091239)
Affinity DataIC50: 1.24E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235604(CHEMBL4088559)
Affinity DataIC50: 1.25E+4nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235604(CHEMBL4088559)
Affinity DataIC50: 1.25E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235623(CHEMBL4064439)
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Mouse)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235605(CHEMBL4094612)
Affinity DataIC50: 1.37E+4nMAssay Description:Antagonist activity at mouse Gal4-fused DBD RORgamma LBD (Pro-261-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235619(CHEMBL4073023)
Affinity DataIC50: 1.43E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235619(CHEMBL4073023)
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235623(CHEMBL4064439)
Affinity DataIC50: 1.70E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235618(CHEMBL4093723)
Affinity DataIC50: 1.75E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235605(CHEMBL4094612)
Affinity DataIC50: 2.11E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235606(CHEMBL4067157)
Affinity DataIC50: 2.23E+4nMAssay Description:Antagonist activity at rat Gal4-fused DBD RORbeta LBD (Pro-205-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235605(CHEMBL4094612)
Affinity DataIC50: 2.60E+4nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed
TargetNuclear receptor ROR-alpha(Human)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50235606(CHEMBL4067157)
Affinity DataIC50: 3.01E+4nMAssay Description:Antagonist activity at human Gal4-fused DBD RORalpha LBD (Pro-211-end) expressed in TRex-CHOK1 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2019
Entry Details Article
PubMed