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16 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design, synthesis of phenstatin/isocombretastatin-oxindole conjugates as antimitotic agents.EBI
Csir-Indian Institute of Chemical Technology
Design, synthesis and evaluation of novel 2-butyl-4-chloroimidazole derived peptidomimetics as Angiotensin Converting Enzyme (ACE) inhibitors.EBI
Csir-Indian Institute of Chemical Technology
Identification of the molecular basis of inhibitor selectivity between the human and streptococcal type I methionine aminopeptidases.EBI
Csir-Indian Institute of Chemical Technology
Synthesis and structure-activity relationships of pyridinyl-1H-1,2,3-triazolyldihydroisoxazoles as potent inhibitors of tubulin polymerization.EBI
Csir-Indian Institute of Chemical Technology
Synthesis and biological evaluation of 4-aza-2,3-dihydropyridophenanthrolines as tubulin polymerization inhibitors.EBI
Csir-Indian Institute of Chemical Technology
Design and green synthesis of 2-(diarylalkyl)aminobenzothiazole derivatives and their dual activities as angiotensin converting enzyme inhibitors and calcium channel blockers.EBI
Csir-Indian Institute of Chemical Technology
Synthesis of thio-heterocyclic analogues from Baylis-Hillman bromides as potent cyclooxygenase-2 inhibitors.EBI
Csir-Indian Institute of Chemical Technology
Synthesis of novel l-rhamnose derived acyclic C-nucleosides with substituted 1,2,3-triazole core as potent sodium-glucose co-transporter (SGLT) inhibitors.EBI
Csir-Indian Institute of Chemical Technology
Synthesis and biological evaluation of new epalrestat analogues as aldose reductase inhibitors (ARIs).EBI
Csir-Indian Institute of Chemical Technology
Design, synthesis and evaluation of novel 2-hydroxypyrrolobenzodiazepine-5,11-dione analogues as potent angiotensin converting enzyme (ACE) inhibitors.EBI
Csir-Indian Institute of Chemical Technology
Design and synthesis of cis-restricted benzimidazole and benzothiazole mimics of combretastatin A-4 as antimitotic agents with apoptosis inducing ability.EBI
Csir-Indian Institute of Chemical Technology
An overview on the synthetic and medicinal perspectives of indenopyrazoles.EBI
Csir-Indian Institute of Chemical Technology
Highly functionalized tetrahydropyridines are cytotoxic and selective inhibitors of human puromycin sensitive aminopeptidase.EBI
Csir-Indian Institute of Chemical Technology
Luotonin-A based quinazolinones cause apoptosis and senescence via HDAC inhibition and activation of tumor suppressor proteins in HeLa cells.EBI
Csir-Indian Institute of Chemical Technology
Synthesis and evaluation of novel triazoles and mannich bases functionalized 1,4-dihydropyridine as angiotensin converting enzyme (ACE) inhibitors.EBI
Csir-Indian Institute of Chemical Technology
Synthesis of DNA interactive C3-trans-cinnamide linked β-carboline conjugates as potential cytotoxic and DNA topoisomerase I inhibitors.EBI
Csir-Indian Institute of Chemical Technology