Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50043973
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449244(CHEMBL3125150)
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM20880(CHEMBL429910 | C-aryl glucoside, 6 | BMS-512148 | ...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM20875(CHEMBL245067 | JMC511145 Compound 1 | 1-(2,4-dihyd...)
Affinity DataIC50: 59nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM20875(CHEMBL245067 | JMC511145 Compound 1 | 1-(2,4-dihyd...)
Affinity DataIC50: 61nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449247(CHEMBL3125147)
Affinity DataIC50: 126nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449242(CHEMBL3125151)
Affinity DataIC50: 135nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449239(CHEMBL3125155)
Affinity DataIC50: 147nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449240(CHEMBL3125154)
Affinity DataIC50: 149nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449252(CHEMBL3125142)
Affinity DataIC50: 150nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449251(CHEMBL3125143)
Affinity DataIC50: 152nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449243(CHEMBL3125152)
Affinity DataIC50: 163nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449248(CHEMBL3125146)
Affinity DataIC50: 175nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449253(CHEMBL3125141)
Affinity DataIC50: 186nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449250(CHEMBL3125144)
Affinity DataIC50: 190nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449241(CHEMBL3125153)
Affinity DataIC50: 214nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449247(CHEMBL3125147)
Affinity DataIC50: 220nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449245(CHEMBL3125149)
Affinity DataIC50: 227nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449249(CHEMBL3125145)
Affinity DataIC50: 257nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449254(CHEMBL3125156)
Affinity DataIC50: 311nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449242(CHEMBL3125151)
Affinity DataIC50: 315nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449239(CHEMBL3125155)
Affinity DataIC50: 315nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449249(CHEMBL3125145)
Affinity DataIC50: 367nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449248(CHEMBL3125146)
Affinity DataIC50: 392nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449246(CHEMBL3125148)
Affinity DataIC50: 434nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449252(CHEMBL3125142)
Affinity DataIC50: 435nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449246(CHEMBL3125148)
Affinity DataIC50: 458nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449243(CHEMBL3125152)
Affinity DataIC50: 467nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449251(CHEMBL3125143)
Affinity DataIC50: 467nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449241(CHEMBL3125153)
Affinity DataIC50: 524nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449250(CHEMBL3125144)
Affinity DataIC50: 528nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449253(CHEMBL3125141)
Affinity DataIC50: 621nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449245(CHEMBL3125149)
Affinity DataIC50: 626nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449254(CHEMBL3125156)
Affinity DataIC50: 629nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Csir-Indian Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449240(CHEMBL3125154)
Affinity DataIC50: 693nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed