TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of wild type human N-terminal His-tagged 12-LOX using arachidonic acid as substrate by UV-Vis spectroscopy analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Compound was tested in vitro for inhibition of 12-LO human plateletMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human platelet 12-lipoxygenase was evaluatedMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human platelet-type 12-lipoxygenaseMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human 12-hLOMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal His6-tagged human platelet 12-LOX using arachidonic acid as substrate by UV-vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:UV-vis cuvette-based assay.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of N-terminal His6-tagged human platelet 12-LOX using arachidonic acid as substrate by UV-vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of His-tagged human platelet 12-lipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:UV-vis cuvette-based assay.More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human 12-hLOMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of N-terminal His6-tagged human platelet 12-LOX using arachidonic acid as substrate by UV-vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:UV-vis cuvette-based assay.More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of N-terminal His6-tagged human platelet 12-LOX using arachidonic acid as substrate by UV-vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:UV-vis cuvette-based assay.More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Assay: Compounds are dissolved in DMSO and diluted to 10 mM concentration in DMSO immediately before IC50 analysis. To determine inhibition of the en...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Reaction buffers used for the lipoxygenase assay were as follows: 25 mM HEPES (pH 7.5), with 0.01% Triton X-100. 1 mM 12-HPETE or 1 mM 15-HPETE stock...More data for this Ligand-Target Pair
Ligand Info
