TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 54nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase acidic protein/Polymerase basic protein 2/RNA-directed RNA polymerase catalytic subunit(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Perugia
Curated by ChEMBL
University of Perugia
Curated by ChEMBL
Affinity DataEC50: 5.80E+3nMAssay Description:Inhibition of RdRP activity in Influenza A virus A/PR/8/34 (H1N1) infected in HEK293T cells co-transfected with NP/PA/PB1/PB2/pPolI-Flu-ffLuc/pRL-SV4...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 2.60nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 0.400nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 0.200nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 0.5nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 2.20E+3nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 4.5nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 5.5nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 70nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase catalytic subunit/Polymerase basic protein 1/Polymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jiaxing Andicon Biotech Co.
US Patent
Jiaxing Andicon Biotech Co.
US Patent
Affinity DataEC50: 1.22nMAssay Description:MDCK cells were seeded in a 96-well cell culture plate, and cultured till cell attachment for later use. The drug was serially 3 times diluted from 2...More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase catalytic subunit/Polymerase basic protein 1/Polymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jiaxing Andicon Biotech Co.
US Patent
Jiaxing Andicon Biotech Co.
US Patent
Affinity DataEC50: 0.600nMAssay Description:MDCK cells were seeded in a 96-well cell culture plate, and cultured till cell attachment for later use. The drug was serially 3 times diluted from 2...More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase catalytic subunit/Polymerase basic protein 1/Polymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jiaxing Andicon Biotech Co.
US Patent
Jiaxing Andicon Biotech Co.
US Patent
Affinity DataEC50: 1.24nMAssay Description:MDCK cells were seeded in a 96-well cell culture plate, and cultured till cell attachment for later use. The drug was serially 3 times diluted from 2...More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase catalytic subunit/Polymerase basic protein 1/Polymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Jiaxing Andicon Biotech Co.
US Patent
Jiaxing Andicon Biotech Co.
US Patent
Affinity DataEC50: 0.680nMAssay Description:MDCK cells were seeded in a 96-well cell culture plate, and cultured till cell attachment for later use. The drug was serially 3 times diluted from 2...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: <3nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Inhibition of PB2 in Influenza A virus (A/Weiss/1943(H1N1)) infected in MDCK cells assessed as reduction in virus induced cell death after 5 days by ...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Binding affinity to full length Influenza A virus PB2 cap-binding domain assessed as dissociation constant incubated for 60 mins by fluorescence pola...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 202nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 145nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 46nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 468nMAssay Description:Binding affinity to recombinant Influenza A virus polymerase PB2 cap-binding domain (318 to 413 residues) assessed as dissociation constant by ITC me...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 1.60E+3nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 6.40E+3nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 580nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding affinity to CM5 immobilized N-terminal His/Sumo tagged Influenza A virus (A/WSN/1933(H1N1)) PB2 CBD (318 to 486 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
