Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 12696
LigandPNGBDBM720548(US20250051345, Example 1)
Affinity DataEC50:  220nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720549(US20250051345, Example 2)
Affinity DataEC50:  61nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720550(US20250051345, Example 3)
Affinity DataEC50:  2.00E+3nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720551(US20250051345, Example 4)
Affinity DataEC50:  2.90E+3nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720552(US20250051345, Example 5)
Affinity DataEC50: >2.60E+3nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720553(US20250051345, Example 6)
Affinity DataEC50:  250nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720554(BayK8644 | US20250051345, Comparative Example 1)
Affinity DataEC50:  21nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720555(RS30124 | US20250051345, Comparative Example 2)
Affinity DataEC50:  450nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720556(CGP028392 | US20250051345, Comparative Example 3)
Affinity DataEC50:  280nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720557(CAS 85825-32-7 | US20250051345, Comparative Exampl...)
Affinity DataEC50:  2.24E+3nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720558(CAS 85825-31-6 | US20250051345, Comparative Exampl...)
Affinity DataEC50:  360nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720559(CAS 92638-18-1 | US20250051345, Comparative Exampl...)
Affinity DataEC50:  510nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
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LigandPNGBDBM720560(US20250051345, Comparative Example 7)
Affinity DataEC50:  930nMAssay Description:Electrophysiological characterization of Cav1.2 activators using Cav1.2-HEK293 (AUX) cell line and QPatch 24 hours prior an electrophysiology experim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent