Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50019978
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625292(CHEMBL5424066)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625291(CHEMBL5422361)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625287(CHEMBL5429506)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625288(CHEMBL5425218)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625294(CHEMBL5397177)
Affinity DataIC50: 11nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625290(CHEMBL5409547)
Affinity DataIC50: 11nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625293(CHEMBL5397122)
Affinity DataIC50: 12nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625298(CHEMBL5422964)
Affinity DataIC50: 13nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625285(CHEMBL5420388)
Affinity DataIC50: 13nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625282(CHEMBL5437464)
Affinity DataIC50: 15nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625284(CHEMBL5429974)
Affinity DataIC50: 18nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 19nMAssay Description:Inhibition of BRD3 BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625286(CHEMBL5393966)
Affinity DataIC50: 24nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 28nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 29nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 43nMAssay Description:Inhibition of BRDT BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 44nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 46nMAssay Description:Inhibition of BRD3 BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 50nMAssay Description:Inhibition of BRD3 BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 57nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 59nMAssay Description:Inhibition of BRDT BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625289(CHEMBL5415106)
Affinity DataIC50: 70nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 79nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625296(CHEMBL5437856)
Affinity DataIC50: 87nMAssay Description:Inhibition of BRDT BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 106nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 111nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625280(CHEMBL5422566)
Affinity DataIC50: 164nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625281(CHEMBL5411832)
Affinity DataIC50: 180nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625297(CHEMBL5415295)
Affinity DataIC50: 194nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 261nMAssay Description:Inhibition of BRD3 BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625279(CHEMBL5406228)
Affinity DataIC50: 365nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 415nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 471nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625283(CHEMBL5407801)
Affinity DataIC50: 482nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625295(CHEMBL5440806)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of BRDT BD1 (unknown origin) using biotinylated H4 peptide as substrate preincubated for 15 mins followed by SA-Tb and GST-XL665 addition ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50625278(CHEMBL5406464)
Affinity DataIC50: 4.89E+3nMAssay Description:Inhibition of human N-terminal 6His-tagged BRD4 BD2 (351 to 457 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells using biotinylated...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed