Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50017825
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605172BDBM50605172(CHEMBL5202921)
Affinity DataKd:  213nMAssay Description:Binding affinity to GFP-fused NLRP3 (unknown origin) expressed in HEK293T cells by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605174BDBM50605174(CHEMBL1164920)
Affinity DataIC50: 810nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605172BDBM50605172(CHEMBL5202921)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605166BDBM50605166(CHEMBL5179667)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605173BDBM50605173(CHEMBL5195047)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155928BDBM50155928(3,4-Methylenedioxyb-Nitrostyrene | CHEMBL596380)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605170BDBM50605170(CHEMBL5174725)
Affinity DataIC50: 9.34E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605168BDBM50605168(CHEMBL5172015)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605167BDBM50605167(CHEMBL5194950)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605169BDBM50605169(CHEMBL5208932)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
School of Pharmacy Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605171BDBM50605171(CHEMBL5178237)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated C57BL/6 mouse bone marrow-derived macrophages assessed as reduction in IL-1beta ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed