Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50003006
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465552(CHEMBL4291641 | US10501466, Example B29)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human WDR5 (22 to 334 residues) assessed as reduction in WRAD-mediated human MLL1 ( 3745 to 3969 residues) H3K4 methylation using human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465585(CHEMBL4279907 | US10501466, Example B11)
Affinity DataIC50: 9.27E+3nMAssay Description:Inhibition of human WDR5 (22 to 334 residues) assessed as reduction in WRAD-mediated human MLL1 ( 3745 to 3969 residues) H3K4 methylation using human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465555(CHEMBL4287817)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human WDR5 (22 to 334 residues) assessed as reduction in WRAD-mediated human MLL1 ( 3745 to 3969 residues) H3K4 methylation using human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465586(CHEMBL4294174 | US10501466, Example B14)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human WDR5 (22 to 334 residues) assessed as reduction in WRAD-mediated human MLL1 ( 3745 to 3969 residues) H3K4 methylation using human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465594(CHEMBL4284408 | US10501466, Example B24)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human WDR5 (22 to 334 residues) assessed as reduction in WRAD-mediated human MLL1 ( 3745 to 3969 residues) H3K4 methylation using human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465552(CHEMBL4291641 | US10501466, Example B29)
Affinity DataKi:  0.902nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465552(CHEMBL4291641 | US10501466, Example B29)
Affinity DataKi: <1nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465585(CHEMBL4279907 | US10501466, Example B11)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465585(CHEMBL4279907 | US10501466, Example B11)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465584(CHEMBL4293572)
Affinity DataKi:  2.80nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465593(CHEMBL4283374)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465555(CHEMBL4287817)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465555(CHEMBL4287817)
Affinity DataKi:  8.40nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465586(CHEMBL4294174 | US10501466, Example B14)
Affinity DataKi:  9.40nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465582(CHEMBL4277864)
Affinity DataKi:  9.90nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465583(CHEMBL4288521)
Affinity DataKi:  13nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465606(CHEMBL4291223)
Affinity DataKi:  16nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465603(CHEMBL4285163)
Affinity DataKi:  21nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465579(CHEMBL4294133)
Affinity DataKi:  23nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465586(CHEMBL4294174 | US10501466, Example B14)
Affinity DataKi:  27nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465554(CHEMBL4286527)
Affinity DataKi:  28nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465604(CHEMBL4283339)
Affinity DataKi:  29nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465602(CHEMBL4278618)
Affinity DataKi:  43nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465581(CHEMBL4292999)
Affinity DataKi:  52nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465594(CHEMBL4284408 | US10501466, Example B24)
Affinity DataKi:  65nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465559(CHEMBL4285902)
Affinity DataKi:  76nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465607(CHEMBL4280428)
Affinity DataKi:  95nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465592(CHEMBL4284733)
Affinity DataKi:  105nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465599(CHEMBL4288724)
Affinity DataKi:  118nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465578(CHEMBL4288010)
Affinity DataKi:  148nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465594(CHEMBL4284408 | US10501466, Example B24)
Affinity DataKi:  182nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465572(CHEMBL4284948)
Affinity DataKi:  184nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465580(CHEMBL4276791)
Affinity DataKi:  185nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465591(CHEMBL4294825)
Affinity DataKi:  219nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465574(CHEMBL4291414)
Affinity DataKi:  473nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465601(CHEMBL4284629)
Affinity DataKi:  480nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465575(CHEMBL4286932)
Affinity DataKi:  503nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465569(CHEMBL4278737)
Affinity DataKi:  665nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465608(CHEMBL4288332)
Affinity DataKi:  690nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465556(CHEMBL4283572)
Affinity DataKi:  924nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465565(CHEMBL4292418)
Affinity DataKi:  1.12E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465576(CHEMBL4276691)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465558(CHEMBL4287245)
Affinity DataKi:  1.38E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465577(CHEMBL4280115)
Affinity DataKi:  1.46E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465557(CHEMBL4281521)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465570(CHEMBL4292147)
Affinity DataKi:  3.13E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465573(CHEMBL4276998)
Affinity DataKi:  3.91E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465600(CHEMBL4295183)
Affinity DataKi:  4.13E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465590(CHEMBL4277278)
Affinity DataKi:  7.21E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50465598(CHEMBL4289405)
Affinity DataKi:  7.54E+3nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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