Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 8100
TargetPlasmepsin II(Plasmodium falciparum)
University of Karachi

LigandPNGBDBM233139(2-Nitrobenzohydrazide | Mr-I-53b)
Affinity DataIC50: 1.00E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Karachi

LigandPNGBDBM233141(1,2-Diphenylhydrazine | Mr-II-10)
Affinity DataIC50: 1.05E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Karachi

LigandPNGBDBM233138(Butanohydrazide | Mr-I-33)
Affinity DataIC50: 1.25E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Karachi

LigandPNGBDBM233139(2-Nitrobenzohydrazide | Mr-I-53b)
Affinity DataIC50: 1.30E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Karachi

LigandPNGBDBM233140(2-Nitrobenzohydrazide | Mr-I-179)
Affinity DataIC50: 1.35E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Karachi

LigandPNGBDBM233138(Butanohydrazide | Mr-I-33)
Affinity DataIC50: 1.40E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Karachi

LigandPNGBDBM233142(1,2-Dipyridinylhydrazine | Mr-II-80)
Affinity DataIC50: 1.45E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Karachi

LigandPNGBDBM50001676(CHEMBL3237776 | Mr-I-27)
Affinity DataIC50: 1.50E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Karachi

LigandPNGBDBM233140(2-Nitrobenzohydrazide | Mr-I-179)
Affinity DataIC50: 1.60E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Karachi

LigandPNGBDBM50001676(CHEMBL3237776 | Mr-I-27)
Affinity DataIC50: 1.65E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Karachi

LigandPNGBDBM233141(1,2-Diphenylhydrazine | Mr-II-10)
Affinity DataIC50: 2.40E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Karachi

LigandPNGBDBM233142(1,2-Dipyridinylhydrazine | Mr-II-80)
Affinity DataIC50: 2.50E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed