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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
TYK2 inhibitors and uses thereofBDB
Nimbus Lakshmi
H3 antagonists containing phenoxypiperidine core structureBDB
Richter Gedeon
Dual inhibitor compounds for use in the treatment of neurodegenerative disorders and alzheimer''s diseaseBDB
Fondazione Istituto Itaiano Di Tecnologia
8-(piperazin-1-yl)-1,2,3,4-tetrahydro-isoquinoline derivativesBDB
Idorsia Pharmaceuticals
Heterocyclic inhibitors of PTPN11BDB
The University of Texas System
Selective targeting of lysosomal cysteine proteases with radiolabeled electrophilic substrate analogs.BDB
University of California San Francisco
Antibiotic sensitization using biphenyl tetrazoles as potent inhibitors of Bacteroides fragilis metallo-beta-lactamase.BDB
Merck Research Laboratories
Splicing factor SF3b as a target of the antitumor natural product pladienolide.BDB
Eisai
Rigid duplex alpha-cyclodextrin reversibly connected with disulfide bonds. Synthesis and inclusion complexes.BDB
Institute of Organic Chemistry and Biochemistry As Cr
 
Thermodynamics of molecular recognition by cyclodextrins. 1. Calorimetric titration of inclusion complexation of naphthalenesulfonates with .alpha.-, .beta.-, and .gamma.-cyclodextrins: enthalpy-entropy compensationBDB
Himeji Institute of Technology
 
Chiral Recognition Thermodynamics of β-Cyclodextrin: The Thermodynamic Origin of Enantioselectivity and the Enthalpy-Entropy Compensation EffectBDB
Japan Science and Technology Agency
Aroylguanidine-based factor Xa inhibitors: the discovery of BMS-344577.BDB
Bristol-Myers Squibb
Discovery of begacestat, a Notch-1-sparing gamma-secretase inhibitor for the treatment of Alzheimer's disease.BDB
Wyeth Research
Structural analysis of ARC-type inhibitor (ARC-1034) binding to protein kinase A catalytic subunit and rational design of bisubstrate analogue inhibitors of basophilic protein kinases.BDB
University of Tartu
Discovery of novel spirocyclopropyl hydroxamate and carboxylate compounds as TACE inhibitors.BDB
Schering-Plough Research Institute
Synthesis and biological evaluation of 4-amino derivatives of benzimidazoquinoxaline, benzimidazoquinoline, and benzopyrazoloquinazoline as potent IKK inhibitors.BDB
Bristol-Myers Squibb