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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and Evaluation of Macrocyclic Peptide Aldehydes as Potent and Selective Inhibitors of the 20S Proteasome.EBI
Whitman College
Protease inhibitors: current status and future prospects.EBI
University of Queensland
D-amino acid containing, high-affinity inhibitors of recombinant human calpain I.EBI
Cephalon
 
Peptidyl aldehyde derivatives as potent and selective inhibitors of cathepsin LEBI
TBA
Molecular modeling: a search for a calpain inhibitor as a new treatment for cataractogenesis.EBI
University of Canterbury
Peptidyl alpha-ketoamides with nucleobases, methylpiperazine, and dimethylaminoalkyl substituents as calpain inhibitors.EBI
Georgia Institute of Technology
Molecular design to enhance the penetration into the retina via ocular instillation.EBI
Senju Pharmaceutical
Exploration of orally available calpain inhibitors 2: peptidyl hemiacetal derivatives.EBI
Senju Pharmaceutical
New peptidic cysteine protease inhibitors derived from the electrophilic alpha-amino acid aziridine-2,3-dicarboxylic acid.EBI
Albert-Ludwigs-University of Freiburg
The role of N-terminal heterocycles in hydrogen bonding to α-chymotrypsin.EBI
The University of Adelaide
Tripeptide analogues of MG132 as protease inhibitors.EBI
University of Adelaide
Novel peptidyl alpha-keto amide inhibitors of calpains and other cysteine proteases.EBI
Georgia Institute of Technology
Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases.EBI
Georgia Institute of Technology
Stereospecific synthesis of peptidyl alpha-keto amides as inhibitors of calpain.EBI
Alkermes
Methods of use of cyclopamine analogsBDB
Infinity Pharmaceuticals
Macrocyclic insulin-degrading enzyme (IDE) inhibitors and uses thereofBDB
President and Fellows of Harvard College