Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50047469
TargetCathepsin B(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50069985({1-[(S)-(S)-1-((S)-1-Formyl-3-methyl-butylcarbamoy...)
Affinity DataKi:  230nMAssay Description:Inhibition of human liver cathepsin B using Cbz-RR-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCalpain-2 catalytic subunit(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50069985({1-[(S)-(S)-1-((S)-1-Formyl-3-methyl-butylcarbamoy...)
Affinity DataKi:  653nMAssay Description:Inhibition of m-calpain (unknown origin) using Suc-LY-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCalpain-2 catalytic subunit(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50169089(CHEMBL3804980)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of m-calpain (unknown origin) using Suc-LY-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCalpain-2 catalytic subunit(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50169088(CHEMBL3806032)
Affinity DataKi:  2.03E+3nMAssay Description:Inhibition of m-calpain (unknown origin) using Suc-LY-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCathepsin B(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50169089(CHEMBL3804980)
Affinity DataKi:  2.29E+3nMAssay Description:Inhibition of human liver cathepsin B using Cbz-RR-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCalpain-2 catalytic subunit(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50169087(CHEMBL3805992)
Affinity DataKi:  2.98E+3nMAssay Description:Inhibition of m-calpain (unknown origin) using Suc-LY-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCathepsin B(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50169088(CHEMBL3806032)
Affinity DataKi:  3.05E+3nMAssay Description:Inhibition of human liver cathepsin B using Cbz-RR-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCathepsin B(Human)
Whitman College

Curated by ChEMBL
LigandPNGBDBM50169087(CHEMBL3805992)
Affinity DataKi:  3.03E+4nMAssay Description:Inhibition of human liver cathepsin B using Cbz-RR-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed