22 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
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[1,2]Oxazolo[5,4-e]isoindoles as promising tubulin polymerization inhibitors.
University of Palermo
Water-soluble isoindolo[2,1-a]quinoxalin-6-imines: in vitro antiproliferative activity and molecular mechanism(s) of action.
University of Palermo
Novel 1H-pyrrolo[2,3-b]pyridine derivative nortopsentin analogues: synthesis and antitumor activity in peritoneal mesothelioma experimental models.
University of Palermo
3D-QSAR pharmacophore modeling and in silico screening of new Bcl-xl inhibitors.
University of Palermo
Identification of 6,9-dihydro-5H-pyrrolo[3,2-h]quinazolines as a new class of F508del-CFTR correctors for the treatment of cystic fibrosis.
University of Palermo
Bioisosteric heterocyclic analogues of natural bioactive flavonoids by scaffold-hopping approaches: State-of-the-art and perspectives in medicinal chemistry.
University of Palermo
1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation.
University of Palermo
Insight into non-nucleoside triazole-based systems as viral polymerases inhibitors.
University of Palermo
Quinoline anticancer agents active on DNA and DNA-interacting proteins: From classical to emerging therapeutic targets.
University of Palermo
Targeting SARS-CoV-2 Main Protease for Treatment of COVID-19: Covalent Inhibitors Structure-Activity Relationship Insights and Evolution Perspectives.
University of Palermo
Synthesis of 2H-Imidazo[2',1':2,3] [1,3]thiazolo[4,5-e]isoindol-8-yl-phenylureas with promising therapeutic features for the treatment of acute myeloid leukemia (AML) with FLT3/ITD mutations.
University of Palermo
Metabolomics-assisted discovery of a new anticancer GLS-1 inhibitor chemotype from a nortopsentin-inspired library: From phenotype screening to target identification.
University of Palermo
Pyrrolomycins as antimicrobial agents. Microwave-assisted organic synthesis and insights into their antimicrobial mechanism of action.
University of Palermo
Synthetic small molecules as anti-biofilm agents in the struggle against antibiotic resistance.
University of Palermo
Synthesis and biological activities of a new class of heat shock protein 90 inhibitors, designed by energy-based pharmacophore virtual screening.
University of Palermo
1,3,5-Triazines: A promising scaffold for anticancer drugs development.
University of Palermo
Synthesis and antitumor activities of 1,2,3-triazines and their benzo- and heterofused derivatives.
University of Palermo
Synthesis, antitumor activity and CDK1 inhibiton of new thiazole nortopsentin analogues.
University of Palermo