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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Crystal structures and pharmacologic activities of 1,4-dihydropyridine calcium channel antagonists of the isobutyl methyl 2,6-dimethyl-4-(substituted phenyl)-1,4-dihydropyridine-3,5-dicarboxylate (nisoldipine) series.EBI
University of Oslo
Synthesis of 5-trifluoromethyl-2-sulfonylpyridine PPARß/d antagonists: Effects on the affinity and selectivity towards PPARß/d.EBI
University of Oslo
Cyclosporine A- and tacrolimus-mediated inhibition of CYP3A4 and CYP3A5 in vitro.EBI
University of Oslo
Synthesis, biological evaluation and molecular modeling studies of the PPARß/d antagonist CC618.EBI
University of Oslo
Synthesis and biological evaluations of new analogs of 2-methoxyestradiol: inhibitors of tubulin and angiogenesis.EBI
University of Oslo
Discovery and pharmacological profile of new hydrophilic 5-HT(4) receptor antagonists.EBI
University of Oslo
Synthesis and evaluation of three structurally related¹8F-labeled orvinols of different intrinsic activities: 6-O-[¹8F]fluoroethyl-diprenorphine ([¹8F]FDPN), 6-O-[¹8F]fluoroethyl-buprenorphine ([¹8F]FBPN), and 6-O-[¹8F]fluoroethyl-phenethyl-orvinol ([¹8F]FPEO).EBI
University of Oslo
Acidic biphenyl derivatives: synthesis and biological activity of a new series of potent 5-HT(4) receptor antagonists.EBI
University of Oslo
Isatin 1,2,3-triazoles as potent inhibitors against caspase-3.EBI
University of Oslo
Synthesis, molecular modeling studies and biological evaluation of fluorine substituted analogs of GW 501516.EBI
University of Oslo
Synthesis of enantiomerically pure milnacipran analogs and inhibition of dopamine, serotonin, and norepinephrine transporters.EBI
University of Oslo
Synthesis and biological evaluations of marine oxohexadecenoic acids: PPARα/γ dual agonism and anti-diabetic target gene effects.EBI
University of Oslo
Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor.EBI
University of Oslo
Molecular modelling, synthesis, and biological evaluations of a 3,5-disubstituted isoxazole fatty acid analogue as a PPARα-selective agonist.EBI
University of Oslo
Synthesis, biological evaluation and molecular modeling of 1,2,3-triazole analogs of combretastatin A-1.EBI
University of Oslo
1,2,3-triazole analogs of combretastatin A-4 as potential microtubule-binding agents.EBI
University of Oslo
1,5-Disubstituted 1,2,3-triazoles as cis-restricted analogues of combretastatin A-4: Synthesis, molecular modeling and evaluation as cytotoxic agents and inhibitors of tubulin.EBI
University of Oslo
Structure-based virtual screening for novel inhibitors of the sarco/endoplasmic reticulum calcium ATPase and their experimental evaluation.BDB
Northern Kentucky University