Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50034250
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  912nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359557(CHEMBL1927476)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359556(CHEMBL1927475)
Affinity DataEC50:  580nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359555(CHEMBL1927474)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359554(CHEMBL1927473)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359557(CHEMBL1927476)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359554(CHEMBL1927473)
Affinity DataEC50:  560nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359556(CHEMBL1927475)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359555(CHEMBL1927474)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359554(CHEMBL1927473)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359557(CHEMBL1927476)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359556(CHEMBL1927475)
Affinity DataEC50:  735nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50359555(CHEMBL1927474)
Affinity DataEC50:  710nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed