49 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Mansoins C-F, Oligomeric Flavonoid Glucosides Isolated from Mansoa hirsuta Fruits with Potential Anti-inflammatory Activity.
University of Mississippi
Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors.
University of Mississippi
1,3,4-Thiadiazoles: a potent multi targeted pharmacological scaffold.
University of Mississippi
Michael acceptor approach to the design of new salvinorin A-based high affinity ligands for the kappa-opioid receptor.
University of Mississippi
Synthesis, biological evaluation, hydration site thermodynamics, and chemical reactivity analysis ofa-keto substituted peptidomimetics for the inhibition of Plasmodium falciparum.
University of Mississippi
Octulosonic acid derivatives from Roman chamomile (Chamaemelum nobile) with activities against inflammation and metabolic disorder.
University of Mississippi
In vitro structure-activity relationships of aplysinopsin analogs and their in vivo evaluation in the chick anxiety-depression model.
University of Mississippi
Structure activity relationship study of benzo[d]thiazol-2(3H)one baseds receptor ligands.
University of Mississippi
Synthesis and evaluation of aplysinopsin analogs as inhibitors of human monoamine oxidase A and B.
University of Mississippi
Glycogen synthase kinase-3 (GSK-3) inhibitory activity and structure-activity relationship (SAR) studies of the manzamine alkaloids. Potential for Alzheimer's disease.
University of Mississippi
Identification of novel parasitic cysteine protease inhibitors using virtual screening. 1. The ChemBridge database.
University of Mississippi
Design and synthesis of the first generation of dithiolane thiazolidinedione- and phenylacetic acid-based PPARgamma agonists.
University of Mississippi
Identification of novel parasitic cysteine protease inhibitors by use of virtual screening. 2. The available chemical directory.
University of Mississippi
Inhibition of human monoamine oxidase A and B by 5-phenoxy 8-aminoquinoline analogs.
University of Mississippi
Synthesis and biological evaluation of new salvinorin A analogues incorporating natural amino acids.
University of Mississippi
Bioassay for the identification of natural product-based activators of peroxisome proliferator-activated receptor-gamma (PPARgamma): the marine sponge metabolite psammaplin A activates PPARgamma and induces apoptosis in human breast tumor cells.
University of Mississippi
Antimalarial (+)-trans-hexahydrodibenzopyran derivatives from Machaerium multiflorum.
University of Mississippi
Cannabinoid Receptor Type II Ligands from Sandalwood Oil and Synthetic α-Santalol Derivatives.
University of Mississippi
A systematic review on the kappa opioid receptor and its ligands: New directions for the treatment of pain, anxiety, depression, and drug abuse.
University of Mississippi
Convenient synthesis and in vitro pharmacological activity of 2-thioanalogs of salvinorins A and B.
University of Mississippi
Isolation and Synthesis of Veranamine, an Antidepressant Lead from the Marine Sponge
University of Mississippi
Kappa-opioid receptor-selective dicarboxylic ester-derived salvinorin A ligands.
University of Mississippi
Semisynthetic studies identify mitochondria poisons from botanical dietary supplements--geranyloxycoumarins from Aegle marmelos.
University of Mississippi
Structures and mechanisms of antitumor agents: xestoquinones uncouple cellular respiration and disrupt HIF signaling in human breast tumor cells.
University of Mississippi
Mitochondrial respiration inhibitors suppress protein translation and hypoxic signaling via the hyperphosphorylation and inactivation of translation initiation factor eIF2α and elongation factor eEF2.
University of Mississippi
Natural and semisynthetic mammea-type isoprenylated dihydroxycoumarins uncouple cellular respiration.
University of Mississippi
Mammea E/BB, an isoprenylated dihydroxycoumarin protonophore that potently uncouples mitochondrial electron transport, disrupts hypoxic signaling in tumor cells.
University of Mississippi
The alternative medicine pawpaw and its acetogenin constituents suppress tumor angiogenesis via the HIF-1/VEGF pathway.
University of Mississippi
Lipophilic 2,5-disubstituted pyrroles from the marine sponge Mycale sp. inhibit mitochondrial respiration and HIF-1 activation.
University of Mississippi
Molecular-targeted antitumor agents. 19. Furospongolide from a marine Lendenfeldia sp. sponge inhibits hypoxia-inducible factor-1 activation in breast tumor cells.
University of Mississippi
Terpenoid tetrahydroisoquinoline alkaloids emetine, klugine, and isocephaeline inhibit the activation of hypoxia-inducible factor-1 in breast tumor cells.
University of Mississippi
Sodwanone and yardenone triterpenes from a South African species of the marine sponge Axinella inhibit hypoxia-inducible factor-1 (HIF-1) activation in both breast and prostate tumor cells.
University of Mississippi
Antimalarial, cytotoxic, and antifungal alkaloids from Duguetia hadrantha.
University of Mississippi
Molecular-targeted antitumor agents: the Saururus cernuus dineolignans manassantin B and 4-O-demethylmanassantin B are potent inhibitors of hypoxia-activated HIF-1.
University of Mississippi
Cytotoxic metabolites from an Indonesian sponge Lendenfeldia sp.
University of Mississippi
Benzochromenones from the marine crinoid Comantheria rotula inhibit hypoxia-inducible factor-1 (HIF-1) in cell-based reporter assays and differentially suppress the growth of certain tumor cell lines.
University of Mississippi
Laurenditerpenol, a new diterpene from the tropical marine alga Laurenciaintricata that potently inhibits HIF-1 mediated hypoxic signaling in breast tumor cells.
University of Mississippi
INHIBITOR OF APOPTOSIS (IAP) PROTEIN ANTAGONISTS
Sanford Burnham Prebys Medical Discovery Institute
Identification of novel p38alpha MAP kinase inhibitors using fragment-based lead generation.
Astex