14 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Synthesis of benzofuran derivatives as selective inhibitors of tissue-nonspecific alkaline phosphatase: effects on cell toxicity and osteoblast-induced mineralization.
University of Lyon
Synthesis and biological evaluation of tetrahydro[1,4]diazepino[1,2-a]indol-1-ones as cyclin-dependent kinase inhibitors.
University of Lyon
Synthesis and biological evaluation of benzo[4,5]imidazo[1,2-c]pyrimidine and benzo[4,5]imidazo[1,2-a]pyrazine derivatives as anaplastic lymphoma kinase inhibitors.
University of Lyon
Inhibitors of tissue-nonspecific alkaline phosphatase: design, synthesis, kinetics, biomineralization and cellular tests.
University of Lyon
Binding evaluation of fragment-based scaffolds for probing allosteric enzymes.
University of Lyon
Synthesis and biological evaluation of potential 5-HT(7) receptor PET radiotracers.
University of Lyon
Synthesis and evaluation of benzo[b]thiophene derivatives as inhibitors of alkaline phosphatases.
University of Lyon
Design of a structure-activity relationship model of vitamin K epoxide reductase (VKORC1) inhibitors combining chemical synthesis of new compounds, enzymatic assays and molecular modelling.
University of Lyon
Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion.
University of Lyon
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of Action.
University of Lyon
New 1-arylindoles based serotonin 5-HT7 antagonists. Synthesis and binding evaluation studies.
University of Lyon
Modular construction of quaternary hemiaminal-based inhibitor candidates and their in cellulo assessment with HIV-1 protease.
University of Lyon