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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design, synthesis, docking studies and biological evaluation of novel dihydro-1,3,5-triazines as human DHFR inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and pharmacological investigation of aralkyl diamine derivatives as potential triple reuptake inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and antidepressant activity of arylalkanol-piperidine derivatives as triple reuptake inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and antidepressant activity of novel 1-(1-benzoylpiperidin-4-yl) methanamine derivatives selectively targeting SSRI/5-HTEBI
Shanghai Institute of Pharmaceutical Industry
Histone deacetylase 6 inhibitors with blood-brain barrier penetration as a potential strategy for CNS-Disorders therapy.EBI
Shanghai Institute of Pharmaceutical Industry
Discovery of potent and selective Bcl-2 inhibitors with acyl sulfonamide skeleton.EBI
Shanghai Institute of Pharmaceutical Industry
Design, synthesis and biological evaluation of brain penetrant benzazepine-based histone deacetylase 6 inhibitors for alleviating stroke-induced brain infarction.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and biological evaluation of novel antipsychotic trans-4-(2-(1,2,4,5-tetrahydro-3H-benzo[d]azepin-3-yl)ethyl)cyclohexan-1-amine derivatives targeting dopamine/serotonin receptor subtypes.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and biological evaluation of novel 1-substituted 3-(3-phenoxyprop-1-yn-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amines as potent Bruton's tyrosine kinase (BTK) inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and antidepressant-like activity of novel aralkyl piperazine derivatives targeting SSRI/5-HTEBI
Shanghai Institute of Pharmaceutical Industry
Design, synthesis and biological evaluation of novel 3-substituted pyrazolopyrimidine derivatives as potent Bruton's tyrosine kinase (BTK) inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and biological evaluation of novel 6,11-dihydro-5H-benzo[e]pyrimido- [5,4-b][1,4]diazepine derivatives as potential c-Met inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Synthesis and antidepressant activity of a series of arylalkanol and aralkyl piperazine derivatives targeting SSRI/5-HTEBI
Shanghai Institute of Pharmaceutical Industry
Design, synthesis and biological evaluation of novel histone deacetylase inhibitors incorporating 4-aminoquinazolinyl systems as capping groups.EBI
Shanghai Institute of Pharmaceutical Industry
1-Acetyl-5-phenyl-1H-pyrrol-3-ylacetate: An aldose reductase inhibitor for the treatment of diabetic nephropathy.EBI
Shanghai Institute of Pharmaceutical Industry
Design, synthesis and biological evaluation of 4-piperazinyl-containing Chidamide derivatives as HDACs inhibitors.EBI
Shanghai Institute of Pharmaceutical Industry
Combination therapy with MDM2 and EFGR inhibitorsBDB
TBA
Interactions of (+)- and (-)-8- and 7-hydroxy-2-(di-n-propylamino)tetralin at human (h)D3, hD2 and h serotonin1A receptors and their modulation of the activity of serotoninergic and dopaminergic neurones in rats.BDB
Institut De Recherches Servier
A-85380 [3-(2(S)-azetidinylmethoxy) pyridine]: in vitro pharmacological properties of a novel, high affinity alpha 4 beta 2 nicotinic acetylcholine receptor ligand.BDB
Abbott Laboratories