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19 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Evaluation of class I HDAC isoform selectivity of largazole analogues.EBI
Duke University
A single step purification for autolytic zinc proteinases.EBI
Duke University
Analysis of HIF-1 inhibition by manassantin A and analogues with modified tetrahydrofuran configurations.EBI
Duke University
Inhibition of Cdc25 phosphatases by indolyldihydroxyquinones.EBI
Duke University
Synthesis and evaluation of cyclopentane-based muraymycin analogs targeting MraY.EBI
Duke University
Inhibition of the antibacterial target UDP-(3-O-acyl)-N-acetylglucosamine deacetylase (LpxC): isoxazoline zinc amidase inhibitors bearing diverse metal binding groups.EBI
Duke University
Structure-Functional-Selectivity Relationship Studies of Novel Apomorphine Analogs to Develop D1R/D2R Biased Ligands.EBI
Duke University
Synthesis and Biological Evaluation of Manassantin Analogues for Hypoxia-Inducible Factor 1α Inhibition.EBI
Duke University
Synthesis, structure, and antibiotic activity of aryl-substituted LpxC inhibitors.EBI
Duke University
Synthesis and biological evaluation of largazole zinc-binding group analogs.EBI
Duke University
Pyrazolopyrimidine compound and preparation method therefor and use thereof in preparation of anti-cancer drugBDB
Suzhou Raymon Pharmaceuticals Company
LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITORS AND USES THEREOFBDB
Insilico Medicine Ip
Selective histone deactylase 6 inhibitorsBDB
H. Lee Moffitt Cancer Center and Research Institute
TRPA1 antagonistsBDB
Abbvie
Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the difference.BDB
Universita Degli Studi Di Firenze
Synthesis of bivalent beta2-adrenergic and adenosine A1 receptor ligands.BDB
Monash University
Discovery of raltegravir, a potent, selective orally bioavailable HIV-integrase inhibitor for the treatment of HIV-AIDS infection.BDB
Merck Research Laboratories
Identification of Inhibitors of Protein Kinase B Using Fragment-Based Lead Discovery.BDB
Astex