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24 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and biological evaluation of a unique heparin mimetic hexasaccharide for structure-activity relationship studies.EBI
Momenta Pharmaceuticals
Improved total synthesis and biological evaluation of potent apratoxin S4 based anticancer agents with differential stability and further enhanced activity.EBI
University of Florida
Bioassay-guided isolation of proanthocyanidins with antiangiogenic activities.EBI
University of Salerno
A focused sulfated glycoconjugate Ugi library for probing heparan sulfate-binding angiogenic growth factors.EBI
The University of Queensland
Synthesis and biological evaluation of polysulfated oligosaccharide glycosides as inhibitors of angiogenesis and tumor growth.EBI
Progen Pharmaceuticals
Discovery of a Dual Tubulin and Neuropilin-1 (NRP1) Inhibitor with Potent In Vivo Anti-Tumor Activity via Pharmacophore-based Docking Screening, Structure Optimization, and Biological Evaluation.EBI
China Pharmaceutical University
Dimer Peptide Ligands of Vascular Endothelial Growth Factor: Optimizing Linker Length for High Affinity and Antiangiogenic Activity.EBI
University Paris Cite
Synthesis, biological activity, and preliminary pharmacokinetic evaluation of analogues of a phosphosulfomannan angiogenesis inhibitor (PI-88).EBI
Progen Industries
1,4-DIHETEROCYCLIC SUBSTITUTED AROMATIC RING OR AROMATIC HETEROCYCLIC COMPOUND AND USE THEREOFBDB
Bebetter Med
PYRIDINO-OR PYRIMIDO-CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOFBDB
Genfleet Therapeutics (Shanghai)
HSD17B13 INHIBITORS AND/OR DEGRADERSBDB
Pfizer
AMPK activatorsBDB
Kallyope
Cyanopyrrolidine derivatives as inhibitors for DUBsBDB
Mission Therapeutics
Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitorsBDB
Boehringer Ingelheim International
Pyrrolidine derivatives and their use as complement pathway modulatorsBDB
Novartis
Quaternized amines as sodium channel blockersBDB
Purdue Pharma
Design, synthesis and SAR study of hydroxychalcone inhibitors of human ß-secretase (BACE1).BDB
Shanghai Institute of Material Medica, Chinese Academy of Sciences
Pyrrolo[3,2-c]pyridine tropomyosin-related kinase inhibitorsBDB
Pfizer
Flap modulatorsBDB
Janssen Pharmaceutica
1′-substituted pyrimidine N-nucleoside analogs for antiviral treatmentBDB
Gilead Sciences
MAPK/ERK kinase inhibitorsBDB
Takeda Pharmaceutical