Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50020588
TargetAtrial natriuretic peptide receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 850nMAssay Description:Inhibition of [125I]-VEGF-A165 binding to NPR1 (unknown origin) transfected in HUVECs incubated for 2 hrs by plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAtrial natriuretic peptide receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50313491((S)-2-(3-(benzo[c][1,2,5]thiadiazole-4-sulfonamido...)
Affinity DataIC50: 2.91E+3nMAssay Description:Inhibition of [125I]-VEGF-A165 binding to NPR1 (unknown origin) transfected in HUVECs incubated for 2 hrs by plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAtrial natriuretic peptide receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631618(CHEMBL5420260)
Affinity DataIC50: 3.91E+3nMAssay Description:Inhibition of [125I]-VEGF-A165 binding to NPR1 (unknown origin) transfected in HUVECs incubated for 2 hrs by plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAtrial natriuretic peptide receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631619(CHEMBL5441104)
Affinity DataIC50: 6.33E+3nMAssay Description:Inhibition of [125I]-VEGF-A165 binding to NPR1 (unknown origin) transfected in HUVECs incubated for 2 hrs by plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAtrial natriuretic peptide receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631620(CHEMBL5403761)
Affinity DataIC50: 8.94E+3nMAssay Description:Inhibition of [125I]-VEGF-A165 binding to NPR1 (unknown origin) transfected in HUVECs incubated for 2 hrs by plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCyclin-G-associated kinase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCyclin-dependent kinase 7(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetTyrosine-protein kinase Fgr(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FGR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ERK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCyclin-dependent kinase 9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 20(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetDual specificity protein kinase TTK(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSTE20-like serine/threonine-protein kinase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SLK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCyclin-dependent kinase 8(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetTyrosine-protein kinase HCK(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HCK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase ICK(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ICK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 8(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JNK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetTyrosine-protein kinase Lck(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LCK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase MAK(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MST1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase 38(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NDR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIK3CA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of RAF1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ROS1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetVascular endothelial growth factor A(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetNeuropilin-2(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NRP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAP2-associated protein kinase 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetActivin receptor type-1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ACVR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetActivin receptor type-2A(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ACVR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAtypical kinase COQ8A, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ADCK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAtypical kinase COQ8B, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ADCK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AKT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AKT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetRAC-gamma serine/threonine-protein kinase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AKT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetALK tyrosine kinase receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ALK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetAnkyrin repeat and protein kinase domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ANKK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetTyrosine-protein kinase Blk(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BLK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BMX (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetCyclin-dependent kinase 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50631617(CHEMBL5440517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
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