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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Vialinin A is a ubiquitin-specific peptidase inhibitor.EBI
Tokyo University of Agriculture
Structure-activity relationship, kinetic mechanism, and selectivity for a new class of ubiquitin C-terminal hydrolase-L1 (UCH-L1) inhibitors.EBI
Harvard Medical School
Mechanisms, biology and inhibitors of deubiquitinating enzymes.EBI
Institute For Bio-Medical Research
Identification of covalent fragment inhibitors for Plasmodium falciparum UCHL3 with anti-malarial efficacy.EBI
Purdue University
Recent advances in the development of ubiquitin-specific-processing protease 7 (USP7) inhibitors.EBI
Zhengzhou University
UCH-L3 structure and function: Insights about a promising drug target.EBI
University of Science and Technology
Activity-based protein profiling reveals deubiquitinase and aldehyde dehydrogenase targets of a cyanopyrrolidine probe.EBI
Imperial College London
Chemical Toolkit for PARK7: Potent, Selective, and High-Throughput.EBI
Leiden University Medical Center
Synthesis and evaluation of tiaprofenic acid-derived UCHL5 deubiquitinase inhibitors.EBI
Wayne State University
Discovery of Potent, Selective, and Orally Bioavailable Inhibitors of USP7 with In Vivo Antitumor Activity.EBI
Rapt Therapeutics
Advances in Discovering Deubiquitinating Enzyme (DUB) Inhibitors.EBI
Dana-Farber Cancer Institute
Chemical Approaches to Intervening in Ubiquitin Specific Protease 7 (USP7) Function for Oncology and Immune Oncology Therapies.EBI
Progenra
INHIBITORS OF BRUTON'S TYROSINE KINASEBDB
Pharmacyclics
Treatment of upper aerodigestive tract disorders and coughBDB
Individual
Ghrelin O-acyltransferase inhibitorsBDB
Glaxosmithkline Intellectual Property Development
Tricyclic rho kinase inhibitorsBDB
Bristol-Myers Squibb
Guanidine compoundBDB
Astellas Pharma
Thyroid receptor ligands. 6. A high affinity "direct antagonist" selective for the thyroid hormone receptor.BDB
Karo Bio