41 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Influence of azide incorporation on binding affinity by small papain inhibitors.
Radboud University Nijmegen
Squaric acid/4-aminoquinoline conjugates: novel potent antiplasmodial agents.
University of Lisbon. Av. Prof. Gama Pinto
Design, synthesis, and optimization of novel epoxide incorporating peptidomimetics as selective calpain inhibitors.
University of Illinois College of Pharmacy
Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis.
University of Milan
Use of papain as a model for the structure-based design of cathepsin K inhibitors: crystal structures of two papain-inhibitor complexes demonstrate binding to S'-subsites.
Smithkline Beecham Pharmaceuticals
Tanshinones as selective and slow-binding inhibitors for SARS-CoV cysteine proteases.
Korea Research Institute of Bioscience and Biotechnology
Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.
University of Florida
Natural polyprenylated benzophenones inhibiting cysteine and serine proteases.
Federal University of Alfenas
Peptidyl beta-homo-aspartals: specific inhibitors of interleukin-1 beta converting enzyme and its homologues (caspases).
Institute For Drug Research
Design, synthesis and biological evaluation of peptidyl-vinylaminophosphonates as novel cysteine protease inhibitors.
National Chemical Laboratory (Csir-Ncl)
Aza vinyl sulfones: synthesis and evaluation as antiplasmodial agents.
University of Lisbon
HLE-inhibitory alkaloids with a polyketide skeleton from the marine-derived fungus Coniothyrium cereale.
University of Bonn
Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB.
National Human Genome Research Institute
Peptidyl epoxides extended in the P' direction as cysteine protease inhibitors: effect on affinity and mechanism of inhibition.
Bar-Ilan University
Isatin compounds as noncovalent SARS coronavirus 3C-like protease inhibitors.
Peking University
Azapeptides structurally based upon inhibitory sites of cystatins as potent and selective inhibitors of cysteine proteases.
University of Gda£?Sk
Discovery, total synthesis, HRV 3C-protease inhibitory activity, and structure-activity relationships of 2-methoxystypandrone and its analogues.
Merck Research Laboratories
Highly tunable thiosulfonates as a novel class of cysteine protease inhibitors with anti-parasitic activity against Schistosoma mansoni.
University of Glasgow
Novel, nonpeptidic cyanamides as potent and reversible inhibitors of human cathepsins K and L.
Merck Frosst Centre For Therapeutic Research
(S)-Thiirancarboxylic acid as a reactive building block for a new class of cysteine protease inhibitors.
University of WüRzburg
Discovery of New Anti-Schistosomal Hits by Integration of QSAR-Based Virtual Screening and High Content Screening.
Universidade Federal De Goi£S
Combinatorial library of serine and cysteine protease inhibitors that interact with both the S and S' binding sites.
Brown University
Potential Anticancer Agents Characterized from Selected Tropical Plants.
The Ohio State University
Mechanistic studies on the inactivation of papain by epoxysuccinyl inhibitors.
University of Wisconsin
Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases.
Georgia Institute of Technology
Nonpeptidic inhibitors of human leukocyte elastase. 2. Design, synthesis, and in vitro activity of a series of 3-amino-6-arylopyridin-2-one trifluoromethyl ketones.
Zeneca Pharmaceuticals Group
Peptidyl alpha-ketoheterocyclic inhibitors of human neutrophil elastase. 3. In vitro and in vivo potency of a series of peptidyl alpha-ketobenzoxazoles.
Zeneca Pharmaceuticals
Isolation of 1-carboxymethylnicotinic acid from the marine sponge anthosigmella cf. raromicrosclera As a cysteine protease inhibitor1
The University of Tokyo
Isolation and structure determination of nostocyclopeptides A1 and A2 from the terrestrial cyanobacterium Nostoc sp. ATCC53789.
University of Hawaii At Manoa
Acid-sensitive latent inhibitors for proteolytic enzymes: synthesis and characterization.
Amherst College
