33 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Full Sequence Amino Acid Scanning of¿-Defensin RTD-1 Yields a Potent Anthrax Lethal Factor Protease Inhibitor.

State University of New York
Probing the S2' Subsite of the Anthrax Toxin Lethal Factor Using Novel N-Alkylated Hydroxamates.

University of Minnesota
Exploring the influence of the protein environment on metal-binding pharmacophores.

University of California
Small molecule inhibitors of anthrax lethal factor toxin.

Microbiotix
D-proline-based peptidomimetic inhibitors of anthrax lethal factor.

TBA
Antidotes to anthrax lethal factor intoxication. Part 3: Evaluation of core structures and further modifications to the C2-side chain.

Panthera Biopharma
Synthesis and biological evaluation of botulinum neurotoxin a protease inhibitors.

Microbiotix
Amiodarone and bepridil inhibit anthrax toxin entry into host cells.

University of California
Inhibitors of anthrax lethal factor based upon N-oleoyldopamine.

Purdue University
Time-dependent botulinum neurotoxin serotype A metalloprotease inhibitors.

Microbiotix
Antidotes to anthrax lethal factor intoxication. Part 2: structural modifications leading to improved in vivo efficacy.

Panthera Biopharma
Identifying chelators for metalloprotein inhibitors using a fragment-based approach.

University of California
Antidotes to anthrax lethal factor intoxication. Part 1: Discovery of potent lethal factor inhibitors with in vivo efficacy.

Panthera Biopharma
In vivo efficacy of beta-cyclodextrin derivatives against anthrax lethal toxin.

National Institute of Allergy and Infectious Diseases
Synthesis and optimization of thiadiazole derivatives as a novel class of substrate competitive c-Jun N-terminal kinase inhibitors.

Institute For Medical Research
Structure-activity relationship studies of a novel series of anthrax lethal factor inhibitors.

Institute For Medical Research
Inhibitors of anthrax lethal factor.

Purdue University
5-Ene-4-thiazolidinones - An efficient tool in medicinal chemistry.

Danylo Halytsky Lviv National Medical University
Hydroxypyrone derivatives in drug discovery: from chelation therapy to rational design of metalloenzyme inhibitors.

Government College Women University
Zinc enzymes in medicinal chemistry.

Hefei University of Technology
In-cell production of a genetically-encoded library based on the θ-defensin RTD-1 using a bacterial expression system.

University of Southern California
Small molecule inhibitors of anthrax edema factor.

Hawaii Biotech
Pyrazole compound

Sumitomo Dainippon Pharma
N2-(3,4-dimethylphenyl)-6-((4-(p-tolyl)piperazin-1-yl)methyl)-1,3,5-triazine-2,4-diamine

Glucox Biotech
Bicyclic heterocycles as FGFR inhibitors

Incyte Holdings
Pyrazolo-pyrrolidin-4-one derivatives and their use in the treatment of disease

Novartis
Multiple kinase pathway inhibitors

Tolero Pharmaceuticals
Substituted pyrido[4,3-d]pyrimidines as Wee-1 inhibitors

Almac Discovery
Structure-activity relationships for 1-phenylbenzimidazoles as selective ATP site inhibitors of the platelet-derived growth factor receptor.

University of Auckland
Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase. 4. 2-Substituted dipyridodiazepinones as potent inhibitors of both wild-type and cysteine-181 HIV-1 reverse transcriptase enzymes.

Boehringer Ingelheim Pharmaceuticals