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28 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structure-activity relationships of benzothiazole GPR35 antagonists.EBI
University of North Carolina At Greensboro
Imidazole-derived agonists for the neurotensin 1 receptor.EBI
Sanford-Burnham Medical Research Institute
Discovery of ML314, a Brain Penetrant Non-Peptidicβ-Arrestin Biased Agonist of the Neurotensin NTR1 Receptor.EBI
Sanford-Burnham Medical Research Institute
6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35.EBI
University of Bonn
8-Benzamidochromen-4-one-2-carboxylic acids: potent and selective agonists for the orphan G protein-coupled receptor GPR35.EBI
University of Bonn
Synthesis and Agonistic Activity at the GPR35 of 5,6-Dihydroxyindole-2-carboxylic Acid Analogues.EBI
TBA
Thieno[3,2-b]thiophene-2-carboxylic acid derivatives as GPR35 agonists.EBI
Corning
Discovery of Natural Phenols as G Protein-Coupled Receptor-35 (GPR35) Agonists.EBI
TBA
Discovery of 2-(4-methylfuran-2(5H)-ylidene)malononitrile and thieno[3,2-b]thiophene-2-carboxylic acid derivatives as G protein-coupled receptor 35 (GPR35) agonists.EBI
Corning
Discovery of a novel GPR35 agonist with high and equipotent species potency for oral treatment of IBD.EBI
University of Chinese Academy of Sciences
Development and Characterization of Fluorescent Probes for the G Protein-Coupled Receptor 35.EBI
Dalian Institute of Chemical Physics
Structure-Activity Relationship Studies of Coumarin-like Diacid Derivatives as Human G Protein-Coupled Receptor-35 (hGPR35) Agonists and a Consequent New Design Principle.EBI
Chinese Academy of Sciences
SAR Studies of EBI
Chinese Academy of Sciences
Discovery of 2H-Chromen-2-one Derivatives as G Protein-Coupled Receptor-35 Agonists.EBI
Dalian Institute of Chemical Physics
SUBSTITUTED PYRIDINE-2,4-DIONE DERIVATIVESBDB
Medshine Discovery
Chemokine receptor modulators and uses thereofBDB
Flx Bio
IRAK4 inhibiting agentsBDB
Biogen Ma
Inhibitors of lysine specific demethylase-1BDB
Celgene Quanticel Research
Polysubstituted pyridine compound, preparation method, use and pharmaceutical compositionBDB
Peking University Founder Group
IDO inhibitorsBDB
Newlink Genetics
Fused pyrimidine compound or salt thereofBDB
Taiho Pharmaceutical
Substituted benzenesulfonamides as sodium channel blockersBDB
Daewoong Pharmaceutical
Benzoxazolone derivatives as acid ceramidase inhibitors, and their use as medicamentsBDB
University of California
New fluorescent 2-phenylindolglyoxylamide derivatives as probes targeting the peripheral-type benzodiazepine receptor: design, synthesis, and biological evaluation.BDB
Universita Di Pisa
Structural basis for dipeptide amide isoform-selective inhibition of neuronal nitric oxide synthase.BDB
University of California Irvine
Indanylacetic acid derivatives carrying 4-thiazolyl-phenoxy tail groups, a new class of potent PPAR alpha/gamma/delta pan agonists: synthesis, structure-activity relationship, and in vivo efficacy.BDB
Bayer Healthcare Pharmaceuticals
In vitro structure-activity relationship and in vivo characterization of 1-(aryl)-3-(4-(amino)benzyl)urea transient receptor potential vanilloid 1 antagonists.BDB
Abbott Laboratories
Crystal structures of multidrug binding protein TtgR in complex with antibiotics and plant antimicrobials.BDB
Imperial College