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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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23 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design and synthesis of selective, dual fatty acid binding protein 4 and 5 inhibitors.EBI
F. Hoffmann-La Roche
Novel fatty acid binding protein 4 (FABP4) inhibitors: virtual screening, synthesis and crystal structure determination.EBI
Chinese Academy of Sciences
Identification and characterization of a small molecule inhibitor of Fatty Acid binding proteins.EBI
University of Minnesota
Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP).EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Truxillic acid monoamides as fatty acid binding protein 5 inhibitors.EBI
Stony Brook University
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review.EBI
Universita degli Studi di Catania
A Real-World Perspective on Molecular Design.EBI
F. Hoffmann-La Roche
NMR structure of a potent small molecule inhibitor bound to human keratinocyte fatty acid-binding protein.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. An update from 2017 to early 2022.EBI
University of Catania
Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target.EBI
Biovitrum
Development of FABP4/5 inhibitors with potential therapeutic effect on type 2 Diabetes Mellitus.EBI
Fudan University
Exploration of Fragment Binding Poses Leading to Efficient Discovery of Highly Potent and Orally Effective Inhibitors of FABP4 for Anti-inflammation.EBI
Chinese Academy of Sciences
Plant-Based Modulators of Endocannabinoid Signaling.EBI
Concordia University Wisconsin
Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor.EBI
Fudan University
SAR studies on truxillic acid mono esters as a new class of antinociceptive agents targeting fatty acid binding proteins.EBI
Stony Brook University
Substituted pyrimidinones as agonists of the APJ receptorBDB
Amgen
Farnesoid X receptor agonists and uses thereofBDB
Metacrine
Synthesis, ß-glucuronidase inhibition and molecular docking studies of hybrid bisindole-thiosemicarbazides analogs.BDB
Universiti Teknologi Mara
Fluoro-substituted 2-aryl-3,5-dicyano-4-indazolyl-6-methyl-1,4-dihydropyridines and uses thereofBDB
Bayer Intellectual Property
Substituted aminopiperidines as dipeptidyl peptidase-IV inhibitors for the treatment of diabetesBDB
Merck Sharp & Dohme
Substrate envelope-designed potent HIV-1 protease inhibitors to avoid drug resistance.BDB
University of Massachusetts
Inhibitors of JAKBDB
Hoffmann-La Roche
Botryllamides and method of inhibiting PGP in a mammal afflicted with cancerBDB
The United States of America, As Represented By The Secretary, Department of Health and Human Services