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22 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity.EBI
University of Eastern Piedmont
Neuroactive and Anti-inflammatory Frankincense Cembranes: A Structure-Activity Study.EBI
University of Eastern Piedmont
Turmeric Sesquiterpenoids: Expeditious Resolution, Comparative Bioactivity, and a New Bicyclic Turmeronoid.EBI
University of Eastern Piedmont
Discovery of non-electrophilic capsaicinoid-type TRPA1 ligands.EBI
University of Eastern Piedmont
Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors.EBI
University of Eastern Piedmont
Synthesis and preliminary evaluation in tumor bearing mice of new (18)F-labeled arylsulfone matrix metalloproteinase inhibitors as tracers for positron emission tomography.EBI
University of Eastern Piedmont
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2.EBI
University of Eastern Piedmont
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene.EBI
University of Eastern Piedmont
Design, synthesis, and biological evaluation of new (2E,6E)-10-(dimethylamino)-3,7-dimethyl-2,6-decadien-1-ol ethers as inhibitors of human and Trypanosoma cruzi oxidosqualene cyclase.EBI
University of Eastern Piedmont
Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): the homovanillyl moiety.EBI
University of Eastern Piedmont
Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors.EBI
University of Eastern Piedmont
The Oxidation of Phytocannabinoids to Cannabinoquinoids.EBI
University of Eastern Piedmont
Triterpenoid Hydroxamates as HIF Prolyl Hydrolase Inhibitors.EBI
University of Eastern Piedmont
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to EBI
University of Eastern Piedmont
Identification of a Strigoterpenoid with Dual Nrf2 and Nf-κB Modulatory Activity.EBI
University of Eastern Piedmont
Dissecting the pharmacophore of curcumin. Which structural element is critical for which action?EBI
University of Eastern Piedmont
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders.EBI
University of Eastern Piedmont
Electrophilic Triterpenoid Enones: A Comparative Thiol-Trapping and Bioactivity Study.EBI
University of Eastern Piedmont
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies.EBI
University of Eastern Piedmont
Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis.EBI
University of Eastern Piedmont
Iodine-Promoted Aromatization of p-Menthane-Type Phytocannabinoids.EBI
University of Eastern Piedmont
The Bibenzyl Canniprene Inhibits the Production of Pro-Inflammatory Eicosanoids and Selectively Accumulates in Some Cannabis sativa Strains.EBI
University of Eastern Piedmont