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47 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of Selective Phosphodiesterase 1 Inhibitors with Memory Enhancing Properties.EBI
Dart Neuroscience
Design and Synthesis of Novel and Selective Phosphodiesterase 2 (PDE2a) Inhibitors for the Treatment of Memory Disorders.EBI
Dart Neuroscience
Macrocyclic Inhibitors of ERK2 Kinase.EBI
Dart Neuroscience
Pyridyl Isonicotinamide Inhibitors of RAF Kinase.EBI
Dart Neuroscience
Pyrazole Inhibitors of GluN2B NMDA Receptor Subunit.EBI
Dart Neuroscience
Quinazoline Carboxamides as Selective Antagonists of Adenosine 2A Receptor.EBI
Dart Neuroscience
Imidazopyridazine Inhibitors of PI3Kß.EBI
Dart Neuroscience
Dihydropteridinone Inhibitors of BRD4.EBI
Dart Neuroscience
Pyridinonaphthyridinone Inhibitors of Type 2 Methionine Aminopeptidase.EBI
Dart Neuroscience
Novel Pyridyloxadiazole Agonists of Sphingosin-1-phosphate.EBI
Dart Neuroscience
Reversible and irreversible small molecule inhibitors of monoamine oxidase B (MAO-B) investigated by biophysical techniques.EBI
Dart Neuroscience
Novel Disubstituted Pyrimidines as Inhibitors of Bruton's Tyrosine Kinase.EBI
Dart Neuroscience
Pyrrolopyridines-quinazolines Inhibitors of PKR-Like ER Kinase.EBI
Dart Neuroscience
Novel azaindazole sulfonamides inhibitors of serum and glucocorticoid regulated kinase.EBI
Dart Neuroscience
Quinalozinones as Inhibitors of Class I PI3K Kinases.EBI
Dart Neuroscience
Pyrrolopyrimidine Analogues as MKNK Inhibitors.EBI
Dart Neuroscience
Combination of novel imidazopyridazine mps-1 kinase inhibitors and bcl-2 family protein inhibitors.EBI
Dart Neuroscience
Pyrazolsulfonamide agonists of oxytocin receptor.EBI
Dart Neuroscience
Triazolo[4,5-d]pyrimidine Derivatives as Inhibitors of GCN2.EBI
Dart Neuroscience
Novel cycloalkenepyrazoles as inhibitors of bub1 kinase.EBI
Dart Neuroscience
Phenyl carboxamide analogues as spleen tyrosine kinase (syk) inhibitors.EBI
Dart Neuroscience
Thiazolocarboxamide Analogues as NAMPT Inhibitors.EBI
Dart Neuroscience
Quinoline Derivatives as 5-HT6 Receptor PET Ligands.EBI
Dart Neuroscience
PDE2 inhibition: potential for the treatment of cognitive disorders.EBI
Dart Neuroscience
Trisubstituted imidazoles as positive modulators of metabotropic glutamate receptor subtype 5.EBI
Dart Neuroscience
Tricyclic Pyrimidines As Inhibitors of DYRK1A/DYRK1B As Potential Treatment for Down's Syndrome or Alzheimer's Disease.EBI
Dart Neuroscience
Novel thiazolobenzodiazepines as inhibitors of histamine h3 receptor.EBI
Dart Neuroscience
Positive allosteric modulators of nicotinic acetylcholine receptor.EBI
Dart Neuroscience
Irreversible inhibitors of cysteine proteases.EBI
Dart Neuroscience
Modulators of the GPR119 Receptor for the Treatment of Metabolic Syndrome.EBI
Dart Neuroscience
Metabolites of the pyrimidine amine preladenant as adenosine a2a receptor antagonists.EBI
Dart Neuroscience
Aminotriazole and Aminotetrazole Inhibitors of LSD1 as Epigenetic Modulators.EBI
Dart Neuroscience
Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties.EBI
Dart Neuroscience
Treatment of Pain with Spirocylic Cyclohexane Derivatives Having Dual Specificity for ORL-1 and μ-Opioid Receptors.EBI
Dart Neuroscience
Diphenylpropane Derivatives as Agonist of PPAR Nuclear Receptors.EBI
Dart Neuroscience
Anabaseine analogues as modulators of nicotinic acetylcholine receptor.EBI
Dart Neuroscience
Imidazopyrazine Derivatives As Inhibitors of mTOR.EBI
Dart Neuroscience
Negative allosteric modulators of metabotropic glutamate receptor subtype.EBI
Dart Neuroscience
Dihydrooxazines As Inhibitors of BACE-1 or BACE-2.EBI
Dart Neuroscience
Novel and selective inhibitors of histone deacetylase: patent highlight.EBI
Dart Neuroscience
Benzenesulfonyl and Benzenesulfonamide as Modulators of the 5-HT6 Receptor: Patent Highlight.EBI
Dart Neuroscience
Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties.EBI
Dart Neuroscience
Indolinone Inhibitors of ENT1 for the Treatment of Schizophrenia.EBI
Dart Neuroscience
CYCLOPIPERIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOFBDB
Shanghaitech University
Bicyclic compounds as ATX inhibitorsBDB
Hoffmann-La Roche
1-cyano-pyrrolidine derivatives as DUB inhibitorsBDB
Mission Therapeutics
Pyridine derivativeBDB
Astellas Pharma