Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50002344
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457379(CHEMBL4211925)
Affinity DataIC50: 14nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457390(CHEMBL4208680)
Affinity DataIC50: 17nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457381(CHEMBL4211194)
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457387(CHEMBL4215413)
Affinity DataIC50: 24nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457386(CHEMBL4212967)
Affinity DataIC50: 26nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457385(CHEMBL4207561)
Affinity DataIC50: 27nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457378(CHEMBL4203736)
Affinity DataIC50: 31nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457384(CHEMBL4210157)
Affinity DataIC50: 39nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457376(CHEMBL4213616)
Affinity DataIC50: 52nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457377(CHEMBL4205790)
Affinity DataIC50: 57nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457388(CHEMBL4217494)
Affinity DataIC50: 97nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457380(CHEMBL4206265)
Affinity DataIC50: 244nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457383(CHEMBL4216732)
Affinity DataIC50: 253nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457382(CHEMBL4213885)
Affinity DataIC50: 321nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457389(CHEMBL4212469)
Affinity DataIC50: 838nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed