15 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors.
Aurigene Discovery Technologies
Discovery of azetidine based ene-amides as potent bacterial enoyl ACP reductase (FabI) inhibitors.
Aurigene Discovery Technologies
Structure-guided discovery of 1,3,5 tri-substituted benzenes as potent and selective matriptase inhibitors exhibiting in vivo antitumor efficacy.
Aurigene Discovery Technologies
Discovery of Pyridyl Bis(oxy)dibenzimidamide Derivatives as Selective Matriptase Inhibitors.
Aurigene Discovery Technologies
Discovery of 7-azaindole based anaplastic lymphoma kinase (ALK) inhibitors: wild type and mutant (L1196M) active compounds with unique binding mode.
Aurigene Discovery Technologies
Design and synthesis of 2-substituted benzoxazoles as novel PTP1B inhibitors.
Aurigene Discovery Technologies
Discovery of MAP855, an Efficacious and Selective MEK1/2 Inhibitor with an ATP-Competitive Mode of Action.
Aurigene Discovery Technologies
Discovery of CA-4948, an Orally Bioavailable IRAK4 Inhibitor for Treatment of Hematologic Malignancies.
Aurigene Discovery Technologies
5-hydroxytryptamine receptor 7 modulators and their use as therapeutic agents
Temple University
Adrenergic receptor modulating compounds and methods of using the same
The Leland Stanford Junior University
Compositions for APP-selective BACE inhibition and uses therefor
University of California
Alkynyl pyridine prolyl hydroxylase inhibitor, and preparation method and medical use thereof
Jiangsu Hengrui Medicine